SCHEMBL8206773

SCHEMBL8206773

CCc1cc(C(=O)NCc2ccccc2)c(N)s1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
ALOX15 P16050 7/20 0.51
LMNA P02545 2/20 0.51
HSD17B10 Q99714 2/20 0.51
KMT2A Q03164 3/20 0.50
NSD2 O96028 2/20 0.50
GAA P10253 3/20 0.49
MAPK1 P28482 2/20 0.49
MEN1 O00255 1/20 0.48
HPGD P15428 3/20 0.48
TP53 P04637 1/20 0.48
GLA P06280 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
POLB P06746 1/20 0.47
ALDH1A1 P00352 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199058 0.87 THRB (0.52) CYP2C19ALOX15LMNAHSD17B10KMT2A
SCHEMBL8211556 0.87 ALOX15 (0.53) ALOX15LMNAHSD17B10KMT2AMEN1
SCHEMBL8210407 0.83 KMT2A (0.53) CYP3A4CYP2C9CYP2C19ALOX15LMNA
SCHEMBL8210426 0.82 ACKR3 (0.53) CYP3A4ALOX15LMNAHSD17B10KMT2A
SCHEMBL8200539 0.81 HSP90AA1 (0.55) CYP3A4CYP2C19LMNAKMT2ANSD2
SCHEMBL8200561 0.80 TAAR1 (0.59) CYP3A4CYP2C9CYP2C19ALOX15LMNA
SCHEMBL20915155 0.80 GAA (0.72) ALOX15HSD17B10KMT2ANSD2GAA
SCHEMBL8207225 0.79 HPGD (0.60) ALOX15LMNAHSD17B10KMT2AMAPK1
SCHEMBL7425279 0.78 NCEH1 (0.46) CYP2C19ALOX15LMNAHSD17B10KMT2A
SCHEMBL8206426 0.78 GAA (0.53) ALOX15LMNAHSD17B10KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed