SCHEMBL8200637

SCHEMBL8200637

CCOC(=O)c1c(C)sc(N)c1C(=O)O

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FHIT P49789 1/20 0.83
ALDH1A1 P00352 14/20 0.68
MAPT P10636 11/20 0.68
HPGD P15428 9/20 0.68
GAA P10253 8/20 0.68
SMN1; SMN2 Q16637 2/20 0.68
TDP1 Q9NUW8 2/20 0.60
RAB9A P51151 3/20 0.58
NPC1 O15118 2/20 0.58
HSD17B10 Q99714 3/20 0.55
ALOX15 P16050 2/20 0.55
MAPK1 P28482 2/20 0.55
KMT2A Q03164 5/20 0.54
MEN1 O00255 4/20 0.54
GRM6 O15303 2/20 0.52
NPSR1 Q6W5P4 1/20 0.52
KDM4E B2RXH2 4/20 0.51
POLB P06746 1/20 0.49
RECQL P46063 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28267388 0.93 FHIT (0.83) FHITALDH1A1MAPTHPGDGAA
SCHEMBL13343389 0.91 FHIT (1.00) FHITALDH1A1MAPTHPGDGAA
SCHEMBL27969857 0.89 ALDH1A1 (0.85) FHITALDH1A1MAPTHPGDGAA
SCHEMBL1622309 0.82 FHIT (0.77) FHITALDH1A1MAPTHPGDGAA
SCHEMBL223094 0.81 ALDH1A1 (1.00) FHITALDH1A1MAPTHPGDGAA
SCHEMBL14708470 0.81 FHIT (0.74) FHITALDH1A1MAPTHPGDGAA
SCHEMBL24811161 0.79 FHIT (0.72) FHITALDH1A1MAPTHPGDGAA
SCHEMBL5119925 0.79 FHIT (0.72) FHITALDH1A1MAPTHPGDGAA
SCHEMBL9097179 0.79 FHIT (0.72) FHITALDH1A1MAPTHPGDGAA
Bromide SCHEMBL28146660 0.79 FHIT (0.51) FHITALDH1A1MAPTHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106749317-B A kind of azepine penthienate [2,3-d] pyrimidone benzsulfamide analog derivative and purposes 中国科学院新疆理化技术研究所 2019-01-01 CN disclosed
WO-2008063668-A1 HETEROBICYCLIC METALLOPROTEASE INHIBITORS ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2008-05-29 WO disclosed