SCHEMBL8200710

SCHEMBL8200710

CC(C)(C)OC(=O)NCCNC(=O)[C@H]1O[C@@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.53
KMT2A Q03164 3/20 0.53
ATM Q13315 3/20 0.53
MEN1 O00255 1/20 0.52
CTSS P25774 3/20 0.50
CTSK P43235 2/20 0.50
MAPK1 P28482 1/20 0.50
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
AKT1 P31749 1/20 0.47
APP P05067 1/20 0.46
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
KLK5 Q9Y337 1/20 0.45
PPARA Q07869 2/20 0.44
PPARG P37231 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200707 1.00 ACE (0.53) ACEKMT2AATMMEN1CTSS
SCHEMBL7205866 0.90 CTSS (0.47) ACEKMT2AATMMEN1CTSS
SCHEMBL7205858 0.90 CTSS (0.47) ACEKMT2AATMMEN1CTSS
SCHEMBL7283491 0.79 ACE (0.61) ACEKMT2AATMCTSSCTSK
SCHEMBL795685 0.79 ACE (0.79) ACEKMT2AATMCTSSCTSK
SCHEMBL21473784 0.79 ACE (0.79) ACEKMT2AATMCTSSCTSK
SCHEMBL606309 0.79 ACE (0.79) ACEKMT2AATMCTSSCTSK
SCHEMBL66220 0.79 ACE (0.79) ACEKMT2AATMCTSSCTSK
SCHEMBL67020 0.79 ACE (0.79) ACEKMT2AATMCTSSCTSK
SCHEMBL27909397 0.79 ACE (0.79) ACEKMT2AATMCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6110967-A USEFUL AS AGENTS FOR PREVENTING AND TREATING METABOLIC OSTEOPATHY SUCH AS OSTEOPOROSIS, HYPERCALCEMIA AND BONE METASTASIS OF CANCER BECAUSE THEY SPECIFICALLY INHIBITS CATHEPSIN L AND ITS FAMILY ENZYMES TO INHIBIT BONE RESORPTION TAIHO PHARMACEUTICALS CO., LTD. (JP) 2000-08-29 US disclosed