SCHEMBL8201130

SCHEMBL8201130

N#CN(Cc1ccc(NS(=O)(=O)c2cccc(C(F)(F)F)c2)cc1)/C(N)=N\c1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
SERPINE1 P05121 1/20 0.45
NAMPT P43490 1/20 0.44
KMT2A Q03164 2/20 0.44
NR3C1 P04150 1/20 0.43
PGR P06401 1/20 0.43
AR P10275 1/20 0.43
ESR2 Q92731 1/20 0.43
HSD17B2 P37059 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
GAA P10253 1/20 0.41
PIK3CB P42338 1/20 0.41
CA2 P00918 1/20 0.40
IDH2 P48735 1/20 0.40
THRB P10828 2/20 0.40
LMNA P02545 1/20 0.40
HSPD1 P10809 2/20 0.40
PTPN2 P17706 2/20 0.40
PTPN1 P18031 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978263 0.83 NAMPT (0.49) TSHRSERPINE1NAMPTKMT2ANR3C1
SCHEMBL8195508 0.81 HTT (0.54) NAMPTKMT2ALMNA
SCHEMBL8195014 0.81 HTT (0.54) NAMPTKMT2ALMNA
SCHEMBL7978261 0.79 NAMPT (0.55) TSHRSERPINE1NAMPTKMT2ANR3C1
SCHEMBL7966282 0.78 GAA (0.43) TSHRNAMPTKMT2AGAALMNA
SCHEMBL8201132 0.75 SERPINE1 (0.54) TSHRSERPINE1NAMPTKMT2ANR3C1
SCHEMBL8200238 0.71 PLG (0.40) TSHRKMT2AGAALMNAMAPT
SCHEMBL8200233 0.70 CYP17A1 (0.45)
SCHEMBL19639260 0.69 NR3C1 (0.55) TSHRSERPINE1NAMPTKMT2ANR3C1
SCHEMBL2689551 0.66 HDAC1 (0.67) TSHRSERPINE1KMT2ANR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000061561-A1 CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO claimed