SCHEMBL8201132

SCHEMBL8201132

N#CNC(=N)N(Cc1ccc(NS(=O)(=O)c2cccc(C(F)(F)F)c2)cc1)c1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 6/20 0.54
NAMPT P43490 2/20 0.49
TSHR P16473 1/20 0.46
HSD17B2 P37059 1/20 0.45
KMT2A Q03164 2/20 0.44
NR3C1 P04150 1/20 0.43
PGR P06401 1/20 0.43
AR P10275 1/20 0.43
ESR2 Q92731 1/20 0.43
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
IDH2 P48735 1/20 0.41
EPHB4 P54760 1/20 0.40
HSPD1 P10809 2/20 0.40
PTPN2 P17706 2/20 0.40
PTPN1 P18031 2/20 0.40
PTPN5 P54829 2/20 0.40
HSPE1 P61604 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978263 0.82 NAMPT (0.49) SERPINE1NAMPTTSHRHSD17B2KMT2A
SCHEMBL8195511 0.81 HTT (0.55) SERPINE1NAMPTKMT2A
SCHEMBL7978261 0.76 NAMPT (0.55) SERPINE1NAMPTTSHRHSD17B2KMT2A
SCHEMBL8201130 0.75 TSHR (0.46) SERPINE1NAMPTTSHRHSD17B2KMT2A
SCHEMBL19639260 0.69 NR3C1 (0.55) SERPINE1NAMPTTSHRHSD17B2KMT2A
SCHEMBL8201250 0.69 CYP17A1 (0.43) NAMPTTSHRKMT2AHDAC1
SCHEMBL12505777 0.67 HDAC6 (0.54) SERPINE1KMT2AHDAC8
SCHEMBL2689551 0.67 HDAC1 (0.67) SERPINE1TSHRHSD17B2KMT2ANR3C1
SCHEMBL7572806 0.66 NR3C1 (0.69) SERPINE1TSHRHSD17B2KMT2ANR3C1
SCHEMBL3558864 0.66 NR3C1 (0.59) SERPINE1TSHRHSD17B2KMT2ANR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000061561-A1 CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO claimed