SCHEMBL8201204

SCHEMBL8201204

COc1ccc(-c2c(C(F)(F)F)n[nH]c2-c2ccc(S(=O)(=O)CCOCCO)cc2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.39
PTGS1 P23219 5/20 0.39
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196703 0.92 PTGS2 (0.42) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8194835 0.90 PTGS2 (0.41) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8187629 0.89 PTGS2 (0.41) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8200043 0.89 PTGS2 (0.40) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8195825 0.88 PTGS2 (0.38) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8195559 0.86 POLB (0.40) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8201303 0.86 PTGS2 (0.43) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8194868 0.86 PTGS2 (0.44) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8196960 0.85 PTGS2 (0.40) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8196083 0.85 ALDH1A1 (0.40) PTGS2PTGS1ALDH1A1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed