SCHEMBL8201677

SCHEMBL8201677

COc1ccc(-c2c[nH]nc2C(F)(F)F)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.44
PTGS1 P23219 3/20 0.43
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
KDM4E B2RXH2 1/20 0.40
KMO O15229 2/20 0.39
GRIN2B Q13224 1/20 0.38
FYN P06241 1/20 0.38
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3480587 0.79 PDK2 (0.49)
SCHEMBL3480536 0.78 CYP11B2 (0.48)
SCHEMBL3480534 0.78 TDP1 (0.39)
SCHEMBL8195793 0.75 IDO1 (0.41) MEN1KMT2A
SCHEMBL17795211 0.74 PDE3B (0.40) PTGS2PTGS1KMO
SCHEMBL21262444 0.73 ENPP1 (0.43) KDM4EMEN1KMT2A
SCHEMBL10554279 0.73 MAPT (0.43) PTGS2PTGS1ADORA2AADORA1KDM4E
SCHEMBL10556563 0.72 PTGS2 (0.47) PTGS2PTGS1ADORA2AADORA1KDM4E
SCHEMBL12326172 0.72 PTGS2 (0.53) PTGS2PTGS1ADORA2AADORA1KMO
SCHEMBL8194882 0.71 PTGS2 (0.38) PTGS2PTGS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed