SCHEMBL10554279

SCHEMBL10554279

COc1ccc(-c2nc(C(F)(F)F)c(Br)[nH]2)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
TP53 P04637 1/20 0.43
THRB P10828 1/20 0.43
PTGS2 P35354 3/20 0.40
PTGS1 P23219 1/20 0.40
KDM4E B2RXH2 2/20 0.40
ENPP3 O14638 2/20 0.39
ENPP1 P22413 2/20 0.39
CHEK2 O96017 2/20 0.39
AMY1A P0DUB6 2/20 0.38
KMO O15229 1/20 0.38
ALOX5 P09917 1/20 0.37
EPHX2 P34913 1/20 0.37
TBK1 Q9UHD2 1/20 0.37
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
PPARG P37231 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10556563 0.74 PTGS2 (0.47) MAPTTP53PTGS2PTGS1KDM4E
SCHEMBL8201677 0.73 PTGS2 (0.44) PTGS2PTGS1KDM4EKMOMEN1
SCHEMBL12326172 0.68 PTGS2 (0.53) PTGS2PTGS1KMOMEN1ALDH1A1
SCHEMBL9217797 0.68 NPBWR1 (0.38) THRBPTGS1KDM4EENPP3ENPP1
SCHEMBL12130381 0.65 KMO (0.44) PTGS2PTGS1KDM4EKMOMEN1
SCHEMBL6002654 0.65 SMPD3 (0.56) MAPTKDM4EKMOALDH1A1ADORA2A
SCHEMBL30096868 0.65 TBK1 (0.42) MAPTTP53THRBKDM4ETBK1
SCHEMBL31305536 0.65 SMPD3 (0.51) MAPTKDM4ECHEK2AMY1AALOX5
SCHEMBL26134931 0.65 SMPD3 (0.51) MAPTKDM4ECHEK2AMY1AALOX5
SCHEMBL8715460 0.65 MAPT (0.49) MAPTTP53THRBPTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4853383-A β-blocking substituted imidazoles MERCK & CO., INC. (US) 1989-08-01 US disclosed
US-4642311-A β-adrenergic blocking imidazolylphenoxy propanolamines MERCK & CO., INC. (US) 1987-02-10 US disclosed