SCHEMBL8201750

SCHEMBL8201750

C=CCCC(C)(C)COC(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)OC)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PEPD P12955 2/20 0.42
FKBP1A P62942 1/20 0.38
XPNPEP1 Q9NQW7 1/20 0.36
CYP3A4 P08684 2/20 0.35
KLK5 Q9Y337 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
ELANE P08246 2/20 0.35
STAT6 P42226 2/20 0.35
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8211908 0.85 PEPD (0.41) PEPDFKBP1AXPNPEP1CYP3A4KLK5
SCHEMBL12055223 0.80 PEPD (0.49) PEPDFKBP1AXPNPEP1KLK5ELANE
SCHEMBL9966624 0.80 PEPD (0.41) PEPDFKBP1AXPNPEP1ELANE
SCHEMBL8246140 0.80 FKBP1A (0.42) FKBP1AELANESTAT6
SCHEMBL8096010 0.78 PEPD (0.41) PEPDFKBP1AXPNPEP1CYP3A4KLK5
SCHEMBL16502012 0.77 PEPD (0.40) PEPDFKBP1AXPNPEP1CYP3A4KLK5
SCHEMBL8227277 0.77 PEPD (0.43) PEPDFKBP1AXPNPEP1CYP3A4KLK5
SCHEMBL14610244 0.77 STAT6 (0.36) PEPDFKBP1ACYP3A4KLK5ALDH1A1
SCHEMBL8046113 0.77 KLK5 (0.51) PEPDFKBP1AXPNPEP1KLK5ELANE
SCHEMBL14202917 0.77 KLK5 (0.51) PEPDFKBP1AXPNPEP1KLK5ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008057209-A1 HCV NS3 PROTEASE INHIBITORS MERCK & CO., INC. (US) 2008-05-15 WO disclosed