SCHEMBL9966624

SCHEMBL9966624

C=CCC(C)(C)COC(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)OC)C(C)C

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PEPD P12955 2/20 0.41
ELANE P08246 8/20 0.40
FKBP1A P62942 1/20 0.38
CMA1 P23946 7/20 0.38
XPNPEP1 Q9NQW7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096010 0.86 PEPD (0.41) PEPDFKBP1AXPNPEP1
SCHEMBL16502012 0.85 PEPD (0.40) PEPDFKBP1AXPNPEP1
SCHEMBL8201750 0.80 PEPD (0.42) PEPDELANEFKBP1AXPNPEP1
SCHEMBL12599485 0.79 CYP3A4 (0.49) PEPDELANEXPNPEP1
SCHEMBL8246560 0.79 FKBP1A (0.43) PEPDFKBP1A
SCHEMBL7316962 0.79 CMA1 (0.51) PEPDELANECMA1XPNPEP1
SCHEMBL8352620 0.79 CMA1 (0.51) PEPDELANECMA1XPNPEP1
SCHEMBL8168154 0.79 CMA1 (0.51) PEPDELANECMA1XPNPEP1
SCHEMBL15692923 0.76 FKBP1A (0.46) PEPDELANEFKBP1AXPNPEP1
SCHEMBL1985159 0.74 ELANE (0.48) ELANECMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082672-A2 PROCESS AND INTERMEDIATES FOR PREPARING MACROLACTAMS MERCK SHARP & DOHME CORP. (US) 2012-06-21 WO disclosed