SCHEMBL8096010

SCHEMBL8096010

C=CCC(C)(C)COC(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)OC)C1CCCC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PEPD P12955 2/20 0.41
FKBP1A P62942 9/20 0.40
XPNPEP1 Q9NQW7 1/20 0.37
KLK5 Q9Y337 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
POLB P06746 2/20 0.35
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
BIRC2 Q13490 2/20 0.33
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16502012 0.99 PEPD (0.40) PEPDFKBP1AXPNPEP1KLK5ALDH1A1
SCHEMBL8246560 0.92 FKBP1A (0.43) PEPDFKBP1AALDH1A1POLB
SCHEMBL9966624 0.86 PEPD (0.41) PEPDFKBP1AXPNPEP1
SCHEMBL8203043 0.81 ALDH1A1 (0.38) ALDH1A1CYP3A4TSHRLMNARAB9A
SCHEMBL731388 0.80 CASP1 (0.36) ALDH1A1CYP3A4TSHRLMNARAB9A
SCHEMBL1244172 0.80 CASP1 (0.36) ALDH1A1CYP3A4TSHRLMNARAB9A
SCHEMBL733205 0.79 CASP1 (0.38) ALDH1A1CYP3A4TSHRLMNARAB9A
SCHEMBL1244162 0.79 CASP1 (0.38) ALDH1A1CYP3A4TSHRLMNARAB9A
SCHEMBL15692746 0.78 PEPD (0.46) PEPDFKBP1AXPNPEP1KLK5ALDH1A1
SCHEMBL23845229 0.78 KLK5 (0.49) PEPDFKBP1AXPNPEP1KLK5POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2178902-B1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2012-11-28 EP disclosed
WO-2009010804-A1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2009-01-22 WO disclosed