SCHEMBL8201875

SCHEMBL8201875

CCc1cc(F)c(C)c2c1NC(=O)CO2

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 5/20 0.39
PARP1 P09874 1/20 0.38
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
DRD2 P14416 3/20 0.35
DRD4 P21917 3/20 0.35
DRD3 P35462 3/20 0.35
MMP12 P39900 1/20 0.35
ADRB1 P08588 7/20 0.34
ADRB2 P07550 5/20 0.34
NR3C1 P04150 2/20 0.33
PGR P06401 2/20 0.33
DRD1 P21728 1/20 0.33
HTR2A P28223 1/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8190736 0.87 PARP1 (0.39) NR3C2PARP1ALDH1A1GAADRD2
SCHEMBL8202568 0.77 RPS6KA1 (0.39) ADRB1ADRB2PDE3BPDE3A
SCHEMBL8198682 0.73 NR3C2 (0.34) NR3C2PARP1ALDH1A1GAADRD2
SCHEMBL14576785 0.72 NR3C2 (0.36) NR3C2ALDH1A1GAADRD2DRD4
SCHEMBL8191321 0.71 MMP12 (0.37) NR3C2ALDH1A1GAADRD2DRD4
SCHEMBL13424803 0.70 PARP1 (0.47) NR3C2PARP1MMP12ADRB1ADRB2
SCHEMBL13369127 0.69 PARP1 (0.56) NR3C2PARP1DRD2DRD3MMP12
SCHEMBL4100343 0.67 DRD2 (0.40) NR3C2ALDH1A1GAADRD2DRD4
SCHEMBL12119317 0.67 DRD2 (0.56) DRD2DRD4DRD3ADRB1ADRB2
SCHEMBL12116980 0.66 PDE3B (0.53) NR3C2PARP1DRD2DRD3MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063668-A1 HETEROBICYCLIC METALLOPROTEASE INHIBITORS ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2008-05-29 WO disclosed