SCHEMBL8201944

SCHEMBL8201944

COc1ccccc1[C@@]1(OC)COCC2(C1)N[C@@H](c1ccc(F)cc1)CO2

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.38
ACHE P22303 3/20 0.33
TSHR P16473 1/20 0.32
HTR7 P34969 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202750 0.90 SLC6A9 (0.32) TACR1ACHE
SCHEMBL8201272 0.87 TACR1 (0.36) TACR1
SCHEMBL8201255 0.87 TACR1 (0.32) TACR1HTR7
SCHEMBL8202155 0.86 TACR1 (0.43) TACR1
SCHEMBL8201838 0.86 SIGMAR1 (0.39) TACR1ACHETSHRHTR2AHTR2C
SCHEMBL8193781 0.74 SLC6A9 (0.36)
SCHEMBL8201159 0.73 TACR1 (0.35) TACR1
SCHEMBL8201999 0.72 GRIN2D (0.36) TACR1ACHESIGMAR1
SCHEMBL8201993 0.72 TACR1 (0.34) TACR1HTR2A
SCHEMBL8202470 0.71 TACR1 (0.38) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080740-A Spiro-ketal derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 2000-06-27 US claimed
US-6080740-A Spiro-ketal derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 2000-06-27 US disclosed