SCHEMBL8201950

SCHEMBL8201950

Cc1c(C(C)C)nc(N)[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.46
PNP P00491 2/20 0.41
NPSR1 Q6W5P4 1/20 0.39
CYP1A2 P05177 1/20 0.39
TYMP P19971 1/20 0.38
MAPT P10636 2/20 0.37
CDK1 P06493 1/20 0.37
CDK4 P11802 1/20 0.37
CDK2 P24941 1/20 0.37
HIF1A Q16665 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
RGS12 O14924 1/20 0.37
LMNA P02545 1/20 0.37
CYP3A4 P08684 1/20 0.37
CASP1 P29466 1/20 0.37
BLM P54132 1/20 0.37
CASP7 P55210 1/20 0.37
GNAI1 P63096 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31727983 0.82 PNP (0.42) XDHPNPNPSR1MAPTCDK1
SCHEMBL8212090 0.80 PNP (0.41) PNPNPSR1CYP1A2MAPTCDK1
SCHEMBL27443358 0.78 KDM4E (0.34) XDHTYMPCDK4KDM4ELMNA
SCHEMBL718210 0.74 NPSR1 (0.52) XDHPNPNPSR1CYP1A2TYMP
SCHEMBL12956972 0.74 CDK1 (0.52) XDHPNPNPSR1CYP1A2TYMP
SCHEMBL14796354 0.72 NPSR1 (0.40) PNPNPSR1HIF1AMEN1KMT2A
SCHEMBL22901877 0.69 PNP (0.45) PNPMAPTHIF1AMITFTP53
SCHEMBL19506131 0.68 XDH (0.46) XDHPNPNPSR1CYP1A2TYMP
SCHEMBL12284639 0.66 ALDH1A1 (0.65) XDHPNPNPSR1CYP1A2MAPT
SCHEMBL22907452 0.65 PNP (0.56) PNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008032171-A1 DIBENZOFURAN DERIVATIVES AS INHIBITORS OF PDE-4 AND PDE-10 MATRIX LABORATORIES LTD. (DE) 2008-03-20 WO disclosed