Biphenyl

Biphenyl

SCHEMBL8201983

C1CNCCN1.c1ccc(-c2ccccc2)cc1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Biphenyl. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.60
HTR1A P08908 2/20 0.50
HTR7 P34969 2/20 0.50
SIGMAR1 Q99720 3/20 0.48
HTR2C P28335 2/20 0.48
CYP1A2 P05177 3/20 0.47
MAPK1 P28482 3/20 0.47
HSD17B10 Q99714 3/20 0.47
CYP3A4 P08684 2/20 0.47
USP2 O75604 2/20 0.47
TP53 P04637 2/20 0.47
CYP2D6 P10635 2/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HTR2A P28223 1/20 0.46
HTR5A P47898 1/20 0.46
HTR6 P50406 1/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biphenyl SCHEMBL27760037 0.97 ALDH1A1 (0.56) ALDH1A1HTR1AHTR7SIGMAR1HTR2C
Biphenyl SCHEMBL27720670 0.97 ALDH1A1 (0.64) ALDH1A1HTR1AHTR7SIGMAR1HTR2C
Biphenyl SCHEMBL28027750 0.91 ALDH1A1 (0.50) ALDH1A1HTR1AHTR7SIGMAR1HTR2C
Biphenyl SCHEMBL3453455 0.88 ALDH1A1 (0.53) ALDH1A1HTR1AHTR7SIGMAR1HTR2C
Biphenyl SCHEMBL28325969 0.87 ALDH1A1 (0.45) ALDH1A1HTR1AHTR7SIGMAR1HTR2C
Biphenyl SCHEMBL10773004 0.85 ALDH1A1 (0.50) ALDH1A1HTR1AHTR7SIGMAR1HTR2C
Piperazine SCHEMBL17065814 0.84 ALDH1A1 (0.71) ALDH1A1HTR1AHTR7SIGMAR1HTR2C
Biphenyl SCHEMBL8466409 0.84 ACP3 (0.47) ALDH1A1HTR1AHTR7SIGMAR1CYP1A2
Biphenyl SCHEMBL28051011 0.84 ALDH1A1 (0.56) ALDH1A1HTR1AHTR7SIGMAR1HTR2C
Biphenyl SCHEMBL29176815 0.83 ALDH1A1 (0.47) ALDH1A1HTR1AHTR7SIGMAR1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 53 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111138713-A Stearylamine modified ammonium polyphosphate and preparation method and application thereof 上海普利特复合材料股份有限公司 2020-05-12 CN claimed
CN-107556255-A A kind of organic amine modified melamine polyphosphate and preparation method thereof 东华大学 2018-01-09 CN claimed
CN-107459492-A A kind of organically-modified melamine polyphosphate and preparation method thereof 东华大学 2017-12-12 CN claimed
CN-117586179-A GPR183 antagonist and synthetic method and application thereof 中国人民解放军海军特色医学中心 2024-02-23 CN disclosed
CN-110498789-B Aralkyl piperidine derivative and application thereof in multi-target anti-depression 上海医药工业研究院 2022-04-05 CN disclosed
US-20220024879-A1 COMPOUNDS FOR TREATMENT OF HEPACI VIRUS INFECTION AND METHOD FOR DETERMINING THERAPY OF HEPACI VIRUS INFECTION, IN PARTICULAR, HCV INFECTION TWINCORE ZENTRUM FUR EXPERIMENTELLE UND KLINISCHE INFEKTIONSFORSCHUNG GMBH (DE) 2022-01-27 US disclosed
CN-110713470-B Flunarizine hydrochloride crystal form B and preparation method thereof 迪嘉药业集团有限公司 2022-01-18 CN disclosed
EP-3898593-A2 COMPOUNDS FOR TREATMENT OF HEPACI VIRUS INFECTION AND METHOD FOR DETERMINING THERAPY OF HEPACI VIRUS INFECTION, IN PARTICULAR, HCV INFECTION Gottfried Wilhelm Leibniz Universität Hannover (DE) 2021-10-27 EP disclosed
CN-112209917-B Application of heterocyclic substituted phenylpiperazine or phenylpiperidine derivatives in antidepressant drugs 上海医药工业研究院 2021-09-24 CN disclosed
CN-112209917-A Application of heterocyclic substituted phenyl piperazine (pyridine) derivatives in antidepressant drugs 上海医药工业研究院 2021-01-12 CN disclosed
WO-2020127211-A2 COMPOUNDS FOR TREATMENT OF HEPACI VIRUS INFECTION AND METHOD FOR DETERMINING THERAPY OF HEPACI VIRUS INFECTION, IN PARTICULAR, HCV INFECTION GOTTFRIED WILHELM LEIBNIZ UNIVERSITÄT HANNOVER (DE) 2020-06-25 WO disclosed
CN-1392140-A Organic compound with bis-4-dicyanomethylene pyran ring and synthetic method and application thereof PHYSICAL & CHEMICAL TECHNOLOGY (CN) 2003-01-22 CN disclosed
CN-1332727-A 3, 3-diarylpiperidine and 2, 2-diarylmorpholine derivatives PFIZER PROD INC (US) 2002-01-23 CN disclosed
EP-1053745-A1 Use of at least a calcium-channel-inhibitor in the treatment of wrinkles L'OREAL (FR) 2000-11-22 EP disclosed
CN-1054850-C Piperazine compounds used in therapy WELLCOME FOUND (GB) 2000-07-26 CN disclosed
CN-1251520-A Use of sodium channel blocker in manfacture of medicament for preventing optic nerve degeneration associated with glaucoma ALLERGAN SALES INC (US) 2000-04-26 CN disclosed
CN-1196732-A Bis-amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors SEARLE & CO (US) 1998-10-21 CN disclosed
CN-1133593-A Piperazine compounds for use in therapy WELLCOME FOUND (GB) 1996-10-16 CN disclosed
US-4309511-A COBALT COMPOUND, COPPER COMPOUND, AND HETEROCYCLIC AMINE AIR PRODUCTS AND CHEMICALS, INC. (US) 1982-01-05 US disclosed
US-3953448-A CORONARY VASODILATION DELMAR CHEMICALS LIMITED (CA) 1976-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220024879-A1 COMPOUNDS FOR TREATMENT OF HEPACI VIRUS INFECTION AND METHOD FOR DETERMINING THERAPY OF HEPACI VIRUS INFECTION, IN PARTICULAR, HCV INFECTION HAVCR2, HCCS, HELZ ALDH1A1 701/4885HTR1A 797/4885HTR7 2532/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.