SCHEMBL8202032

SCHEMBL8202032

CN(C)C(=O)C(C(N)=O)c1cscn1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
HRH1 P35367 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6161752 0.77 KDM4E (0.34) KDM4EALDH1A1TSHR
SCHEMBL2522189 0.75 KDM4E (0.38) KDM4EALDH1A1TSHRHRH1KCNH2
SCHEMBL3160945 0.68 KDM4E (0.35) KDM4EALDH1A1TSHRHRH1KCNH2
SCHEMBL7280997 0.68 KDM4E (0.35) KDM4EALDH1A1TSHR
SCHEMBL1617758 0.68 DPP4 (0.45) KCNH2
SCHEMBL1617776 0.68 DPP4 (0.45) KCNH2
SCHEMBL2926049 0.68
Hydrochloric Acid SCHEMBL6165347 0.67 DPP4 (0.44) KCNH2
Hydrochloric Acid SCHEMBL6165352 0.67 DPP4 (0.44) KCNH2
SCHEMBL3842916 0.67 KDM4E (0.34) KDM4EALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6107329-A HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS PFIZER, INC. (US) 2000-08-22 US disclosed
WO-1996039384-A1 SUBSTITUTED N-(INDOLE-2-CARBONYL)-GLYCINAMIDES AND DERIVATIVES AS GLYCOGEN PHOSPHORYLASE INHIBITORS PFIZER, INC. (US) 1996-12-12 WO disclosed