SCHEMBL8202680

SCHEMBL8202680

COCc1cc(NN)ccc1N

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.33
TDP1 Q9NUW8 3/20 0.33
RECQL P46063 2/20 0.33
ALOX15 P16050 2/20 0.33
CYP3A4 P08684 2/20 0.33
THRB P10828 2/20 0.33
HIF1A Q16665 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 3/20 0.32
KDM4E B2RXH2 2/20 0.32
HPGD P15428 2/20 0.32
MAPT P10636 5/20 0.32
PRKCE Q02156 2/20 0.32
MYLK Q15746 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
PRKCG P05129 1/20 0.32
PRKCA P17252 1/20 0.32
APEX1 P27695 1/20 0.32
TSHR P16473 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10883526 0.76 ALDH1A1 (0.48) ALDH1A1TDP1RECQLALOX15CYP3A4
SCHEMBL19899827 0.76 MAPT (0.44) ALDH1A1TDP1RECQLCYP3A4LMNA
SCHEMBL108757 0.76 MAPT (0.44) ALDH1A1TDP1RECQLCYP3A4LMNA
SCHEMBL29354986 0.76 MAPT (0.44) ALDH1A1TDP1RECQLCYP3A4LMNA
SCHEMBL10248422 0.76 ALDH1A1 (0.39) ALDH1A1CYP3A4GAAKDM4EHPGD
Hydrochloric Acid SCHEMBL552122 0.75 ALDH1A1 (0.38) ALDH1A1CYP3A4GAAKDM4EHPGD
SCHEMBL8099008 0.75 HSD17B3 (0.44) ALDH1A1TDP1RECQLALOX15CYP3A4
Hydrochloric Acid SCHEMBL7132484 0.75 MAPT (0.42) ALDH1A1TDP1RECQLCYP3A4THRB
Hydrochloric Acid SCHEMBL6256039 0.75 MAPT (0.42) ALDH1A1TDP1RECQLCYP3A4THRB
Bromide SCHEMBL26108834 0.75 MAPT (0.42) ALDH1A1TDP1RECQLCYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008053300-A1 PYRAZOLINE COMPOUNDS AS MINERALOCORTICOID RECEPTOR ANTAGONISTS PFIZER PRODUCTS INC. (US) 2008-05-08 WO disclosed