SCHEMBL8203124

SCHEMBL8203124

C=C(NOC(C)OCC(C)C)c1ccc(N2CCC(CNCC3CCC(CN[C@H](C(=O)O)C4CCCCC4)CC3)CC2)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.34
HDAC8 Q9BY41 3/20 0.34
KDM4E B2RXH2 3/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GFER P55789 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ADRB2 P07550 2/20 0.33
ADRB1 P08588 2/20 0.33
ADRB3 P13945 2/20 0.33
MMP13 P45452 1/20 0.31
ADRA1D P25100 2/20 0.31
ADRA1A P35348 2/20 0.31
ADRA1B P35368 2/20 0.31
SMYD3 Q9H7B4 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM1A O60341 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195753 0.92 HDAC3 (0.38) HDAC3HDAC8KDM4EMEN1ALDH1A1
SCHEMBL8205561 0.91 ITGB3 (0.37) HDAC3HDAC8KDM4EMEN1ALDH1A1
SCHEMBL8207131 0.91 ITGB3 (0.32) HDAC3HDAC8KDM4EMEN1ALDH1A1
SCHEMBL13007355 0.89 HDAC3 (0.40) HDAC3HDAC8KDM4EMEN1ALDH1A1
SCHEMBL8212256 0.87 HDAC3 (0.41) HDAC3HDAC8KDM4EMEN1ALDH1A1
SCHEMBL8195555 0.83 KDM4E (0.40) HDAC3HDAC8KDM4EMEN1ALDH1A1
SCHEMBL8206345 0.83 HDAC6 (0.40) HDAC3HDAC8KDM4EADRB2ADRB1
SCHEMBL13007366 0.83 HDAC3 (0.36) HDAC3HDAC8KDM4EMEN1ALDH1A1
SCHEMBL8204583 0.82 OPRM1 (0.34) HDAC3HDAC8HDAC6F10
SCHEMBL8195710 0.81 HDAC6 (0.40) HDAC3HDAC8KDM1AHDAC6FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008053131-A1 HYDROXAMATES AS INHIBITORS OF HISTONE DEACETYLASE CHROMA THERAPEUTICS LTD. (GB) 2008-05-08 WO disclosed