SCHEMBL8203245

SCHEMBL8203245

CCc1ccccc1-c1cc(-c2ccc(C3=NCCN3)cc2)no1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 5/20 0.48
MAOB P27338 11/20 0.47
MAOA P21397 8/20 0.47
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
HPGD P15428 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
HSD17B10 Q99714 1/20 0.45
S1PR1 P21453 1/20 0.43
TOP2A P11388 2/20 0.43
TOP2B Q02880 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8214278 0.80 ALDH1A1 (0.65) NISCHMAOBMAOAALDH1A1CYP1A2
SCHEMBL1794747 0.80 TOP2A (0.61) NISCHMAOBMAOAALDH1A1CYP1A2
SCHEMBL8201663 0.80 CYP1A2 (0.52) NISCHMAOBMAOAALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL1795721 0.79 TOP2A (0.62) NISCHMAOBMAOAALDH1A1CYP1A2
SCHEMBL8201404 0.77 NISCH (0.56) NISCHMAOBMAOAALDH1A1CYP1A2
SCHEMBL1796041 0.77 NISCH (0.56) NISCHMAOBMAOAALDH1A1CYP1A2
SCHEMBL8211455 0.77 NISCH (0.65) NISCHMAOBMAOAALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL1796884 0.76 NISCH (0.55) NISCHMAOBMAOAALDH1A1CYP1A2
SCHEMBL8188588 0.74 LMNA (0.63) NISCHMAOBMAOAALDH1A1CYP1A2
SCHEMBL1795198 0.74 NISCH (0.56) NISCHMAOBMAOAALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000078726-A1 IMIDAZOLINE DERIVATIVES FOR THE TREATMENT OF DIABETES, ESPECIALLY TYPE II DIABETES ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed