SCHEMBL8203929

SCHEMBL8203929

O=C(Oc1cccs1)C1CCCCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.49
KMT2A Q03164 4/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
ELANE P08246 1/20 0.48
HPGD P15428 4/20 0.47
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.43
TSHR P16473 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198206 0.98 KMT2A (0.50) POLBKMT2AHTTSMN1; SMN2TDP1
SCHEMBL8319487 0.95 KMT2A (0.55) POLBKMT2AHTTSMN1; SMN2TDP1
SCHEMBL27318954 0.91 SMN1; SMN2 (0.44) POLBKMT2AHTTSMN1; SMN2TDP1
Hydrochloric Acid SCHEMBL27383606 0.83 MMP1 (0.41) POLBKMT2AHTTSMN1; SMN2TDP1
SCHEMBL6597161 0.78 EPHX1 (0.42) KMT2AHPGDRAB9AMEN1TSHR
SCHEMBL28194803 0.76 HPGD (0.44) POLBKMT2AHPGDRAB9AMEN1
SCHEMBL7271802 0.75 MMP1 (0.40) ELANETSHRCYP1A2CYP3A4CYP2D6
SCHEMBL3122718 0.75 MMP1 (0.40) ELANETSHRCYP1A2CYP3A4CYP2D6
SCHEMBL4594986 0.75 ALDH1A1 (0.39) POLBKMT2AHPGDRAB9AMEN1
SCHEMBL27707429 0.73 MMP1 (0.41) POLBKMT2ASMN1; SMN2HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147051-A ANTIISCHEMIC AGENT TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2000-11-14 US disclosed
EP-0552417-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-07-07 EP disclosed
US-5883075-A HYPOTENSIVE AGENT CYCLIC PEPTIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-03-16 US disclosed
EP-0528312-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-07-16 EP disclosed
US-5616684-A CYCLIC HEXAPEPTIDE CONTAINING ASPARTIC ACID AND DERIVATIVES, 2-THIENYLGLYCINE, LEUCINE, AND TRYPTOPHAN; ENDOTHELIN RECEPTOR ANTAGONIST TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-01 US disclosed
EP-0626174-A2 Methods and compositions for the prophylactic and/or therapeutic treatment of organ hypofunction TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-11-30 EP disclosed
EP-0552417-A1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-07-28 EP disclosed
EP-0528312-A2 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-02-24 EP disclosed