SCHEMBL820467

SCHEMBL820467

CCC(O)C(N)=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354435 1.00
SCHEMBL2325910 1.00
Hydrochloric Acid SCHEMBL2413368 0.97
Methylamine SCHEMBL27403434 0.97 CA1 (0.41)
SCHEMBL8097160 0.85 MAPT (0.36)
SCHEMBL5583603 0.82 ALOX15 (0.34)
SCHEMBL15648928 0.82 EPHX1 (0.34)
Hydrochloric Acid SCHEMBL15648597 0.80 GNAI3 (0.34)
SCHEMBL294878 0.78
SCHEMBL4107937 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 353 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12344618-B2 Heterotricyclic derivative compound and use of same HANMI PHARMACEUTICAL CO., LTD. (KR) 2025-07-01 US claimed
CN-115991666-B Production method of methyl pyrrolidone 中国石油化工股份有限公司 2025-04-25 CN claimed
CN-118994046-A Preparation method of bemat and application of bemat in tablet 重庆圣华曦药业股份有限公司 2024-11-22 CN claimed
CN-118440551-A Long-acting aging-resistant acrylic acid anti-corrosion paint and production process thereof 易元(迁安)新材料科技有限公司 2024-08-06 CN claimed
CN-113423710-B Novel heterocyclic tricyclic derivative compounds and use thereof 韩美药品株式会社 2024-06-14 CN claimed
CN-116964048-A Bicyclic tetrahydroazepine derivatives for the treatment of cancer 豪夫迈·罗氏有限公司 2023-10-27 CN claimed
WO-2023201270-A2 THERAPEUTIC APPLICATIONS OF CRISPR TYPE V SYSTEMS CARIBOU BIOSCIENCES, INC. (US) 2023-10-19 WO claimed
CN-115991666-A Production method of methyl pyrrolidone 中国石油化工股份有限公司 2023-04-21 CN claimed
US-20220135582-A1 NOVEL HETEROTRICYCLIC DERIVATIVE COMPOUND AND USE OF SAME HANMI PHARMACEUTICAL CO., LTD. (KR) 2022-05-05 US claimed
EP-3929199-A1 NOVEL HETEROTRICYCLIC DERIVATIVE COMPOUND AND USE OF SAME Hanmi Pharmaceutical Co., Ltd. (KR) 2021-12-29 EP claimed
WO-2001046131-A1 METHOD FOR MAKING 24(S)-HYDROXYVITAMIN D¿2? BONE CARE INTERNATIONAL, INC. (US) 2001-06-28 WO claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
EP-0972066-A1 ENZYMATIC CONVERSION OF $g(a)-HYDROXYNITRILES TO THE CORRESPONDING $g(a)-HYDROXYAMIDES, ACIDS OR ACID SALTS Novus International, Inc. (US) 2000-01-19 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-5866379-A Enzymatic conversion of α-hydroxynitriles to the corresponding .alpha. NOVUS INTERNATIONAL (US) 1999-02-02 US claimed
WO-1998032872-A1 ENZYMATIC CONVERSION OF α-HYDROXYNITRILES TO THE CORRESPONDING α-HYDROXYAMIDES, ACIDS OR ACID SALTS NOVUS INTERNATIONAL, INC. (US) 1998-07-30 WO claimed
WO-1996003874-A1 ACARICIDAL COMPOSITION PIERRE FABRE SANTE (FR) 1996-02-15 WO claimed
US-4464539-A FROM ALPHAHYDROXY AMIDES USING PHOSPHATE CATALYSTS MITSUI TOATSU CHEMICALS, INC. (JP) 1984-08-07 US claimed
US-4143159-A SKIN-CARE AGENTS CONTAINING HYDROXYALKYL CARBOXAMIDES AND PROCESS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1979-03-06 US claimed
US-4055590-A FROM AN AMIDE AND ALCOHOL, CATALYST ROHM GMBH (DT) 1977-10-25 US claimed