SCHEMBL8204767

SCHEMBL8204767

C[Si](C)(C)c1ccc2c(c1)C(=O)C(=O)C2

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.47
CES1 P23141 1/20 0.47
METAP1 P53582 4/20 0.40
CES2 O00748 4/20 0.33
MIF P14174 1/20 0.33
MAOA P21397 2/20 0.32
TNF P01375 2/20 0.32
ACHE P22303 1/20 0.31
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4899752 0.80 MAPT (0.35) METAP1MAOAACHE
SCHEMBL1512741 0.75 METAP1 (0.67) BCHECES1METAP1MAOAACHE
SCHEMBL12879668 0.73
SCHEMBL4900031 0.71 RAB9A (0.42) MAOAACHE
SCHEMBL8206319 0.71 TDP1 (0.55) BCHECES1METAP1MAOAMAOB
SCHEMBL31638281 0.71 CES1 (0.52) BCHECES1METAP1MAOAMAOB
SCHEMBL26073771 0.71 BCHE (0.52) BCHECES1METAP1MAOAACHE
SCHEMBL8217231 0.70 BCHE (0.47) BCHECES1METAP1CES2MAOA
SCHEMBL1512575 0.70 METAP1 (0.70) BCHECES1METAP1CES2MIF
SCHEMBL1512594 0.70 ALDH1A1 (0.50) BCHECES1METAP1MAOAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127189-A CONTACTING WITH A 1,2-INDANEDIONE DERIVATIVE, MEASURING ABSORBANCE OR FLUORESCENCE OF PRODUCT FORMED, AND COMPARING TO STANDARDS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2000-10-03 US claimed
WO-1998020344-A1 COMPOSITIONS AND METHODS FOR DETECTION OF AN AMINE COMPOUND THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-05-14 WO claimed
US-6127189-A CONTACTING WITH A 1,2-INDANEDIONE DERIVATIVE, MEASURING ABSORBANCE OR FLUORESCENCE OF PRODUCT FORMED, AND COMPARING TO STANDARDS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2000-10-03 US disclosed
WO-1998020344-A1 COMPOSITIONS AND METHODS FOR DETECTION OF AN AMINE COMPOUND THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-05-14 WO disclosed