SCHEMBL8205180

SCHEMBL8205180

Cc1c(Cl)nc(NCC2CCC2)c(=O)n1CC(=O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 11/20 0.52
F2 P00734 2/20 0.44
F7 P08709 1/20 0.44
F3 P13726 1/20 0.44
PRSS1 P07477 1/20 0.44
GPBAR1 Q8TDU6 1/20 0.41
TSHR P16473 1/20 0.41
GRIN2B Q13224 2/20 0.41
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
PLAU P00749 1/20 0.40
ITGB3 P05106 1/20 0.40
ITGAV P06756 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7023919 0.88 TPSAB1 (0.47) TPSAB1F2F7F3PRSS1
SCHEMBL7694668 0.88 TPSAB1 (0.47) TPSAB1F2F7F3PRSS1
SCHEMBL7403728 0.87 TPSAB1 (0.49) TPSAB1F2F7F3PRSS1
SCHEMBL7020326 0.86 TPSAB1 (0.43) TPSAB1F2F7F3PRSS1
SCHEMBL7027708 0.86 TPSAB1 (0.43) TPSAB1F2F7F3PRSS1
SCHEMBL7020466 0.86 TPSAB1 (0.43) TPSAB1F2F7F3PRSS1
SCHEMBL7029085 0.86 TPSAB1 (0.43) TPSAB1F2F7F3PRSS1
SCHEMBL7018545 0.86 TPSAB1 (0.43) TPSAB1F2F7F3PRSS1
SCHEMBL7021799 0.85 TPSAB1 (0.43) TPSAB1F2F7F3PRSS1
SCHEMBL7026301 0.85 TSHR (0.43) TPSAB1F2F7F3PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6011038-A Pyrazinone thrombin inhibitors MERCK & CO., INC. (US) 2000-01-04 US disclosed