SCHEMBL8205397

SCHEMBL8205397

COC(=O)Cc1n[nH]c2c(F)c(F)ccc12

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.53
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.39
P2RX7 Q99572 2/20 0.38
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35
EGFR P00533 2/20 0.35
CDK1 P06493 1/20 0.34
CDK2 P24941 1/20 0.34
GSK3B P49841 1/20 0.34
PPARG P37231 1/20 0.33
NCOA2 Q15596 1/20 0.33
NCOA1 Q15788 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8219414 0.80 SMN1; SMN2 (0.49) SMN1; SMN2MAPTALDH1A1P2RX7KDM4E
SCHEMBL14158476 0.76 P2RX7 (0.39) P2RX7
SCHEMBL22267604 0.72 GSK3B (0.55) SMN1; SMN2MAPTEGFRGSK3BRXFP1
SCHEMBL1377394 0.71 GSK3B (0.58) CDK1CDK2GSK3B
SCHEMBL4300704 0.71 SMN1; SMN2 (0.71) SMN1; SMN2MAPTALDH1A1KDM4EHSD17B10
SCHEMBL14564361 0.70 SMN1; SMN2 (0.55) SMN1; SMN2MAPTALDH1A1KDM4EGSK3B
SCHEMBL9328808 0.70 SMN1; SMN2 (1.00) SMN1; SMN2MAPTALDH1A1KDM4E
SCHEMBL9323964 0.69 SMN1; SMN2 (0.53) SMN1; SMN2MAPTALDH1A1EGFRGSK3B
SCHEMBL6016609 0.69 SMN1; SMN2 (0.53) SMN1; SMN2MAPTALDH1A1GSK3B
SCHEMBL23914767 0.69 MAP2K4 (0.51) SMN1; SMN2MAPTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008040995-A9 INDAZOLES FOR USE AS DPP-IV INHIBITORS PEAKDALE MOLECULAR LTD (GB) 2008-12-31 WO disclosed
WO-2008040995-A1 INDAZOLES FOR USE AS DPP-IV INHIBITORS PEAKDALE MOLECULAR LIMITED (GB) 2008-04-10 WO disclosed