SCHEMBL8207782

SCHEMBL8207782

CC(C)NC(=O)c1cccc(C(=O)NCc2ccc(-c3ccc(N)cc3)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
ROCK2 O75116 1/20 0.47
ROCK1 Q13464 1/20 0.47
KLKB1 P03952 1/20 0.47
KLK1 P06870 1/20 0.47
HPGD P15428 3/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPK8 P45983 2/20 0.45
MAPK9 P45984 2/20 0.45
MAPK10 P53779 2/20 0.45
STAT3 P40763 1/20 0.43
EPHX2 P34913 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
GALR3 O60755 1/20 0.42
NR2F2 P24468 1/20 0.42
PDE2A O00408 1/20 0.42
PPID Q08752 1/20 0.42
HIF1A Q16665 1/20 0.42
PPARA Q07869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8212242 0.91 ROCK2 (0.52) CA1CA2ROCK2ROCK1KLKB1
SCHEMBL8207800 0.91 ROCK2 (0.47) CA1CA2ROCK2ROCK1KLKB1
SCHEMBL8200906 0.90 HPGD (0.54) CA1CA2ROCK2ROCK1HPGD
SCHEMBL8205692 0.88 MAPK8 (0.47) CA1CA2ROCK2ROCK1KLKB1
SCHEMBL8212034 0.88 ROCK2 (0.47) ROCK2ROCK1KLKB1KLK1
SCHEMBL12853369 0.85 XDH (0.49) CA1CA2ROCK2ROCK1HPGD
SCHEMBL8207563 0.85 MAPK8 (0.56) CA1CA2MAPK8MAPK9MAPK10
SCHEMBL29333050 0.85 SMN1; SMN2 (0.51) CA1CA2HPGDALDH1A1SMN1; SMN2
SCHEMBL8198502 0.84 SMN1; SMN2 (0.53) CA1CA2HPGDALDH1A1SMN1; SMN2
SCHEMBL8211821 0.82 ROCK2 (0.47) CA1CA2ROCK2ROCK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008082487-A2 NOVEL JNK INHIBITORS SCHERING CORPORATION (US) 2008-07-10 WO disclosed