SCHEMBL8206685

SCHEMBL8206685

CONC(=O)c1cc(O)cc(C)c1NC(=O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 3/20 0.52
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
MAOA P21397 3/20 0.51
SMN1; SMN2 Q16637 1/20 0.46
POLB P06746 1/20 0.45
MGLL Q99685 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM1A O60341 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28564954 0.85 NPC1 (0.64) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL8207158 0.84 NPC1 (0.54) CASP3NPC1RAB9APOLBMGLL
SCHEMBL8206774 0.83 CASP3 (0.47) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL8197914 0.78 TACR3 (0.55) CASP3NPC1RAB9ATP53MAPT
SCHEMBL16088310 0.77 NPC1 (0.61) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL3041603 0.75 NPC1 (0.58) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL4201818 0.74 NPC1 (0.57) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL6929631 0.74 NPC1 (0.63) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL15720647 0.73 CA12 (0.63) NPC1RAB9ASMN1; SMN2POLBMGLL
SCHEMBL17997751 0.73 NPC1 (0.58) CASP3NPC1RAB9AMAOASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS Takeda Chemical Industries, Ltd. (JP) 2000-02-16 EP disclosed
WO-1998047882-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-29 WO disclosed