SCHEMBL8206774

SCHEMBL8206774

CONC(=O)c1cc(OCCCc2ccccc2)cc(C)c1NC(=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.47
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAOA P21397 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
RECQL P46063 1/20 0.42
MCL1 Q07820 2/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
BLK P51451 1/20 0.40
BTK Q06187 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8206685 0.83 CASP3 (0.52) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL8205935 0.74 SIRT2 (0.50) NPC1RAB9AMAOAMCL1SIRT2
SCHEMBL8197914 0.73 TACR3 (0.55) CASP3NPC1RAB9ATP53MAPT
SCHEMBL8207158 0.73 NPC1 (0.54) CASP3NPC1RAB9AL3MBTL1
SCHEMBL6191271 0.71 NPC1 (0.45) CASP3NPC1RAB9ASMN1; SMN2RECQL
SCHEMBL16088310 0.71 NPC1 (0.61) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL28564954 0.71 NPC1 (0.64) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL4201818 0.68 NPC1 (0.57) CASP3NPC1RAB9AMAOASMN1; SMN2
SCHEMBL7659684 0.68 CASP3 (0.46) CASP3NPC1RAB9ASMN1; SMN2RECQL
SCHEMBL6929631 0.68 NPC1 (0.63) CASP3NPC1RAB9AMAOASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS Takeda Chemical Industries, Ltd. (JP) 2000-02-16 EP disclosed
WO-1998047882-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-29 WO disclosed