SCHEMBL8206801

SCHEMBL8206801

CCn1cccc1-c1cccc(O)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 8/20 0.44
HSD17B1 P14061 7/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP17A1 P05093 2/20 0.40
FYN P06241 4/20 0.39
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2B6 P20813 1/20 0.38
CYP2C19 P33261 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
BAZ2B Q9UIF8 1/20 0.37
BAZ2A Q9UIF9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7034429 0.76 ESR1 (0.41) CYP3A4ESR1
SCHEMBL1501838 0.76 IDO1 (0.53) HSD17B2HSD17B1CYP17A1FYNMKNK1
Propane SCHEMBL5843489 0.72 HSD17B1 (0.71) HSD17B2HSD17B1CYP3A4CYP2C9CYP17A1
Alcohol SCHEMBL9461730 0.71 HSD17B1 (0.68) HSD17B2HSD17B1CYP3A4CYP2C9CYP17A1
SCHEMBL22006701 0.70 ADRA1A (0.35)
Alcohol SCHEMBL23879308 0.69 HSD17B1 (0.65) HSD17B2HSD17B1CYP3A4CYP2C9CYP17A1
SCHEMBL27593555 0.68 PCSK9 (0.40) CYP2C9CYP1A2CYP2C19
Pentane SCHEMBL28008463 0.67 HSD17B1 (0.62) HSD17B2HSD17B1CYP3A4CYP2C9CYP17A1
Propane SCHEMBL27565820 0.67 HSD17B1 (0.70) HSD17B2HSD17B1CYP3A4CYP2C9CYP17A1
Alcohol SCHEMBL23879306 0.67 HSD17B1 (0.62) HSD17B2HSD17B1CYP3A4CYP2C9CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986560-A1 PYRROLO 2,1,5-CD]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES NOVO NORDISK A/S (DK) 2000-03-22 EP claimed
WO-1998055482-A1 PYRROLO[2,1,5-CD]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES NOVO NORDISK A/S (DK) 1998-12-10 WO claimed
EP-0986560-A1 PYRROLO 2,1,5-CD]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES NOVO NORDISK A/S (DK) 2000-03-22 EP disclosed
WO-1998055482-A1 PYRROLO[2,1,5-CD]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES NOVO NORDISK A/S (DK) 1998-12-10 WO disclosed