SCHEMBL8207010

SCHEMBL8207010

NC(=O)C(c1ccccc1)(c1ccccc1)C1CCC(NCCc2cccnc2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
TAAR1 Q96RJ0 1/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
C3AR1 Q16581 2/20 0.38
CYP1A2 P05177 3/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 3/20 0.38
CYP2C19 P33261 2/20 0.38
RECQL P46063 1/20 0.38
HIF1A Q16665 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199053 0.89 TAAR1 (0.50) CHRM2CHRM1CHRM3TAAR1MEN1
SCHEMBL8206393 0.89 TAAR1 (0.43) CHRM2CHRM1CHRM3TAAR1ROCK2
SCHEMBL8199243 0.83 GRIN2B (0.46) TAAR1SIGMAR1
SCHEMBL8206923 0.83 TAAR1 (0.54) TAAR1MEN1KMT2ANPC1RAB9A
SCHEMBL8206646 0.82 TACR1 (0.42) CHRM2CHRM1CHRM3TAAR1MEN1
SCHEMBL8206100 0.81 HSD11B1 (0.42) CHRM2CHRM1CHRM3MEN1KMT2A
Hydrochloric Acid SCHEMBL8209834 0.81 GRIN2B (0.46) TAAR1SIGMAR1
SCHEMBL8207099 0.79 KDM4E (0.46) CHRM2CHRM1CHRM3MEN1KMT2A
SCHEMBL8207012 0.78 KDM4E (0.47) CHRM2CHRM1CHRM3CYP1A2CYP3A4
SCHEMBL8208907 0.78 CHRM2 (0.40) CHRM2CHRM1CHRM3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0999205-A1 AMINOCYCLOALKANE COMPOUNDS Mitsubishi-Tokyo Pharmaceuticals, Inc. (JP) 2000-05-10 EP disclosed