SCHEMBL8207012

SCHEMBL8207012

CN(Cc1cccnc1)C1CCC(C(C(N)=O)(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.43
OPRK1 P41145 1/20 0.42
RIPK1 Q13546 1/20 0.40
FNTA P49354 2/20 0.39
FNTB P49356 2/20 0.39
CHRM2 P08172 2/20 0.39
DHODH Q02127 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
AGTR2 P50052 1/20 0.38
GRM2 Q14416 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
UBE2M P61081 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199055 0.89 AGTR2 (0.43) OPRK1CHRM2CHRM4AGTR2OPRM1
SCHEMBL8206397 0.89 AGTR2 (0.38) ALDH1A1OPRK1FNTAFNTBCHRM2
SCHEMBL8206924 0.84 AGTR2 (0.43) ALDH1A1OPRK1CHRM2CHRM4AGTR2
SCHEMBL8206641 0.82 SLC6A4 (0.40) ALDH1A1OPRK1CHRM2CHRM4AGTR2
SCHEMBL8206102 0.81 MCHR1 (0.41) KDM4EALDH1A1OPRK1CHRM2AGTR2
SCHEMBL8199247 0.81 AGTR2 (0.42) OPRK1CHRM2CHRM4AGTR2OPRM1
SCHEMBL8207101 0.80 CHRM2 (0.46) ALDH1A1CHRM2GRM2OPRM1CHRM1
Hydrochloric Acid SCHEMBL8209836 0.79 AGTR2 (0.47) OPRK1AGTR2OPRM1
SCHEMBL8206406 0.78 UBE2M (0.40) KDM4EALDH1A1OPRK1CHRM2CHRM4
SCHEMBL8207010 0.78 CHRM2 (0.41) ALDH1A1LMNACHRM2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0999205-A1 AMINOCYCLOALKANE COMPOUNDS Mitsubishi-Tokyo Pharmaceuticals, Inc. (JP) 2000-05-10 EP disclosed