SCHEMBL8207520

SCHEMBL8207520

O=C(Oc1cccs1)C(c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.50
TDP1 Q9NUW8 1/20 0.44
POLB P06746 1/20 0.43
CYP2D6 P10635 3/20 0.42
ALDH1A1 P00352 3/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP12 P39900 1/20 0.42
CHRM1 P11229 4/20 0.41
CHRM3 P20309 4/20 0.41
CHRM2 P08172 3/20 0.41
CHRM4 P08173 3/20 0.41
KLK7 P49862 2/20 0.41
CYP1A2 P05177 2/20 0.40
LMNA P02545 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202887 0.83 HPGD (0.47) POLBALDH1A1CYP2C9MMP1MMP2
SCHEMBL8818944 0.83 HPGD (0.47) POLBALDH1A1CYP2C9MMP1MMP2
SCHEMBL8228297 0.77 MMP1 (0.45) TDP1ALDH1A1CYP2C9CYP2C19MMP1
SCHEMBL10670691 0.76 SLC1A3 (0.42) L3MBTL1POLBALDH1A1CYP2C9CYP2C19
SCHEMBL1036006 0.75
SCHEMBL27458824 0.75 MMP1 (0.44) L3MBTL1TDP1ALDH1A1CYP2C9CYP2C19
SCHEMBL27603109 0.74 TRPM8 (0.47) L3MBTL1POLBALDH1A1CYP2C19MMP1
SCHEMBL3399442 0.74 MMP1 (0.43) TDP1POLBALDH1A1MMP1MMP2
SCHEMBL28311881 0.74 MMP1 (0.43) TDP1ALDH1A1CYP2C9MMP1MMP2
SCHEMBL41616 0.74 MMP1 (0.43) TDP1POLBALDH1A1MMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147051-A ANTIISCHEMIC AGENT TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2000-11-14 US disclosed
EP-0552417-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-07-07 EP disclosed
US-5883075-A HYPOTENSIVE AGENT CYCLIC PEPTIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-03-16 US disclosed
EP-0528312-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-07-16 EP disclosed
US-5616684-A CYCLIC HEXAPEPTIDE CONTAINING ASPARTIC ACID AND DERIVATIVES, 2-THIENYLGLYCINE, LEUCINE, AND TRYPTOPHAN; ENDOTHELIN RECEPTOR ANTAGONIST TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-01 US disclosed
EP-0626174-A2 Methods and compositions for the prophylactic and/or therapeutic treatment of organ hypofunction TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-11-30 EP disclosed
EP-0552417-A1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-07-28 EP disclosed
EP-0528312-A2 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-02-24 EP disclosed