SCHEMBL8202887

SCHEMBL8202887

CC(C(=O)Oc1cccs1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.47
PTGS2 P35354 5/20 0.43
PTGS1 P23219 4/20 0.43
CYP2C9 P11712 2/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
KDM4E B2RXH2 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
PKM P14618 1/20 0.41
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
MMP12 P39900 1/20 0.40
KMT2A Q03164 1/20 0.40
FAAH O00519 1/20 0.39
BCHE P06276 1/20 0.38
HTR1A P08908 1/20 0.38
ADRB3 P13945 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8818944 1.00 HPGD (0.47) HPGDPTGS2PTGS1CYP2C9ALDH1A1
SCHEMBL8207520 0.83 L3MBTL1 (0.50) CYP2C9ALDH1A1LMNAPKMMMP1
SCHEMBL11666585 0.83 PTGS2 (0.55) HPGDPTGS2PTGS1CYP2C9LMNA
SCHEMBL28147524 0.82 ALOX5 (0.47) HPGDPTGS2PTGS1CYP2C9ALDH1A1
SCHEMBL8228297 0.81 MMP1 (0.45) HPGDPTGS2PTGS1CYP2C9ALDH1A1
SCHEMBL27458824 0.80 MMP1 (0.44) HPGDPTGS2PTGS1CYP2C9ALDH1A1
SCHEMBL27686399 0.79 PTGS1 (0.43) HPGDPTGS2PTGS1ALDH1A1LMNA
SCHEMBL28311881 0.78 MMP1 (0.43) HPGDPTGS2PTGS1CYP2C9ALDH1A1
SCHEMBL3399442 0.78 MMP1 (0.43) HPGDALDH1A1KDM4EMMP1MMP2
SCHEMBL41616 0.78 MMP1 (0.43) HPGDALDH1A1KDM4EMMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103351318-A Preparation method of 2-(3-carboxymethyl-4-thiophenyl-phenyl) propionic acid CHANGZHOU INST ENG TECH 2013-10-16 CN disclosed
US-6147051-A ANTIISCHEMIC AGENT TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2000-11-14 US disclosed
EP-0552417-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-07-07 EP disclosed
US-5883075-A HYPOTENSIVE AGENT CYCLIC PEPTIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-03-16 US disclosed
EP-0528312-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-07-16 EP disclosed
US-5616684-A CYCLIC HEXAPEPTIDE CONTAINING ASPARTIC ACID AND DERIVATIVES, 2-THIENYLGLYCINE, LEUCINE, AND TRYPTOPHAN; ENDOTHELIN RECEPTOR ANTAGONIST TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-01 US disclosed
EP-0626174-A2 Methods and compositions for the prophylactic and/or therapeutic treatment of organ hypofunction TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-11-30 EP disclosed
EP-0552417-A1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-07-28 EP disclosed
EP-0528312-A2 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-02-24 EP disclosed