SCHEMBL8208914

SCHEMBL8208914

CC(=O)Nc1ccc(-c2ccc(C(=O)C[N+](=O)[O-])cc2)c(Cl)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 5/20 0.37
TP53 P04637 1/20 0.37
HIF1A Q16665 1/20 0.37
MAPT P10636 6/20 0.36
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
USP2 O75604 1/20 0.33
HTT P42858 1/20 0.33
CYP19A1 P11511 1/20 0.32
PDE7A Q13946 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8211884 0.92 KMT2A (0.40) KMT2AALDH1A1TP53HIF1AMAPT
SCHEMBL8215758 0.87 KMT2A (0.35) KMT2AALDH1A1TP53HIF1AMAPT
SCHEMBL8211436 0.80 ALDH1A1 (0.45) KMT2AALDH1A1TP53HIF1AMAPT
SCHEMBL7091629 0.80 CYP2C19 (0.38) ALDH1A1MAPTNPC1POLBRAB9A
SCHEMBL8752484 0.74 ALDH1A1 (0.60) KMT2AALDH1A1TP53HIF1AMAPT
SCHEMBL9640825 0.74 KDM4E (0.61) KMT2AALDH1A1TP53HIF1AMAPT
SCHEMBL7085464 0.73 CYP2C19 (0.41) KMT2AALDH1A1NPC1POLBRAB9A
SCHEMBL6998722 0.72 ADORA2B (0.43) KMT2AMAPTNPC1POLBRAB9A
SCHEMBL7088791 0.71 KMT2A (0.37) KMT2AALDH1A1NPC1POLBRAB9A
SCHEMBL9386214 0.69 GSK3B (0.55) KMT2AALDH1A1MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0983226-A1 NEW NITROMETHYL KETONES, PROCESS FOR PREPARING THEM AND COMPOSITIONS CONTAINING THEM MERCK PATENT GmbH (DE) 2000-03-08 EP claimed
WO-1998052906-A1 NEW NITROMETHYL KETONES, PROCESS FOR PREPARING THEM AND COMPOSITIONS CONTAINING THEM MERCK PATENT GMBH (DE) 1998-11-26 WO claimed