SCHEMBL8209728

SCHEMBL8209728

Cc1ccc(CCCNC2CCC(C(C(N)=O)(c3ccccc3)c3ccccc3)C2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.42
KCNH2 Q12809 1/20 0.41
GRIN2B Q13224 8/20 0.39
SIGMAR1 Q99720 3/20 0.39
GRIN1 Q05586 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM3 P20309 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39
CCR2 P41597 1/20 0.39
PLAAT3 P53816 1/20 0.38
PLAAT5 Q96KN8 1/20 0.38
PLAAT2 Q9NWW9 1/20 0.38
PLAAT4 Q9UL19 1/20 0.38
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199243 0.92 GRIN2B (0.46) GRIN2BSIGMAR1GRIN1OPRM1OPRL1
SCHEMBL8205354 0.91 MEN1 (0.43) GRIN2BSIGMAR1GRIN1ALDH1A1OPRM1
SCHEMBL8199188 0.91 GRIN2B (0.40) KCNH2GRIN2BSIGMAR1GRIN1CHRM2
SCHEMBL8205279 0.90 GRIN2B (0.48) GRIN2BGRIN1ALDH1A1CYP1A2CYP3A4
SCHEMBL8199090 0.90 GRIN2B (0.43) GRIN2BSIGMAR1GRIN1ALDH1A1CHRM2
SCHEMBL8211310 0.89 OPRM1 (0.39) KCNH2GRIN2BSIGMAR1GRIN1CHRM2
Hydrochloric Acid SCHEMBL8209834 0.88 GRIN2B (0.46) GRIN2BSIGMAR1GRIN1OPRM1OPRL1
SCHEMBL8211721 0.88 MCHR1 (0.44) GRIN2BSIGMAR1GRIN1ALDH1A1CYP1A2
SCHEMBL8206072 0.86 GRIN2B (0.48) GRIN2BSIGMAR1ALDH1A1CYP1A2CYP2C9
SCHEMBL8205244 0.86 TAAR1 (0.49) GRIN2BSIGMAR1GRIN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0999205-A1 AMINOCYCLOALKANE COMPOUNDS Mitsubishi-Tokyo Pharmaceuticals, Inc. (JP) 2000-05-10 EP claimed
EP-0999205-A1 AMINOCYCLOALKANE COMPOUNDS Mitsubishi-Tokyo Pharmaceuticals, Inc. (JP) 2000-05-10 EP disclosed