SCHEMBL8209866

SCHEMBL8209866

COCc1cccc(CC=O)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.46
FFAR1 O14842 1/20 0.40
IDO1 P14902 4/20 0.39
AGXT P21549 2/20 0.39
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MIF P14174 1/20 0.37
KDM1A O60341 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
F2 P00734 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL487468 0.85 IDO1 (0.48) ERN1FFAR1IDO1AGXTMAOB
SCHEMBL6600052 0.83 ERN1 (0.43) ERN1FFAR1IDO1AGXTMAOA
SCHEMBL12345478 0.82 MAOB (0.39) MAOAMAOBLMNA
SCHEMBL23478010 0.82 ALDH1A1 (0.50) ERN1ALDH1A1SMN1; SMN2LMNATP53
SCHEMBL28831709 0.81 IDO1 (0.44) ERN1FFAR1IDO1AGXTF2
SCHEMBL12345479 0.81 CHRM2 (0.40) ALDH1A1
SCHEMBL14230490 0.79 ERN1 (0.42) ERN1IDO1AGXTMAOAMAOB
SCHEMBL30800165 0.78 MAOA (0.55) ERN1MAOAMAOBALDH1A1SMN1; SMN2
SCHEMBL1279762 0.78 MAOA (0.55) ERN1MAOAMAOBALDH1A1SMN1; SMN2
SCHEMBL7930766 0.77 MGLL (0.44) IDO1ALDH1A1SMN1; SMN2LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6093812-A LACTAMIZATION OF A 2-HYDROXYALKYLAMIDE IN AQUEOUS SOLUTION BY TREATMENT WITH A POLYCHLOROBENZOYL CHLORIDE, BASE AND PHASE TRANSFER AGENT SCHERING CORPORATION (US) 2000-07-25 US disclosed
US-5561227-A CHLORINATION A CARBOXYLIC ACID; DEPROTONATION A CHIRAL (OXA OR THIA)ZOLIDINONE; ENOLIZING; CYCLIZATION SCHERING CORPORATION (US) 1996-10-01 US disclosed
US-5306817-A Multistep; cyclizing a hydroxyamide by treating with a dialkylchlorophosphate either a metal hydride, or an aqueous solution of base and a phase transfer catalyst SCHERING CORPORATION (US) 1994-04-26 US disclosed