SCHEMBL8212352

SCHEMBL8212352

COC(=O)C1CCC(C(=O)Nc2sc3c(c2C(=O)NCc2ccc(OC)c(Cl)c2)CCCC3)CC1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.55
CNR1 P21554 1/20 0.55
MAPT P10636 8/20 0.52
KDM4E B2RXH2 4/20 0.52
HSD17B10 Q99714 1/20 0.52
MGAM O43451 4/20 0.52
AMY1A P0DUB6 2/20 0.52
ALDH1A1 P00352 3/20 0.50
HPGD P15428 3/20 0.50
POLB P06746 2/20 0.50
LMNA P02545 2/20 0.49
TP53 P04637 3/20 0.48
GAA P10253 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NPSR1 Q6W5P4 1/20 0.47
FLT3 P36888 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7888443 0.94 CNR2 (0.54) CNR2CNR1MAPTKDM4EHSD17B10
Bicarbonate SCHEMBL7426152 0.92 CNR2 (0.59) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL8207571 0.92 CNR2 (0.58) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL7430283 0.86 CNR2 (0.57) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL8206909 0.85 RORC (0.63) CNR2CNR1MAPTKDM4EHSD17B10
Bicarbonate SCHEMBL7430289 0.84 CNR2 (0.62) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL8212606 0.84 CNR2 (0.61) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL8206341 0.83 CNR2 (0.55) CNR2CNR1MAPTKDM4EHSD17B10
SCHEMBL7425023 0.83 KDM4E (0.60) MAPTKDM4EMGAMAMY1AALDH1A1
SCHEMBL8199918 0.83 MGAM (0.64) MAPTKDM4EMGAMAMY1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed