SCHEMBL8214342

SCHEMBL8214342

Fc1ccc(Cl)cc1NBr

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.40
CCR2 P41597 3/20 0.39
KMT2A Q03164 3/20 0.38
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.38
KCNMA1 Q12791 3/20 0.38
GRM4 Q14833 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
NPC1 O15118 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
P2RX1 P51575 1/20 0.36
P2RX4 Q99571 1/20 0.36
P2RX7 Q99572 1/20 0.36
FLT1 P17948 1/20 0.36
KCNN3 Q9UGI6 1/20 0.36
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29669311 0.84 KMT2A (0.47) CCR2KMT2ALMNATAS1R3TAS1R1
SCHEMBL9231470 0.81 GAA (0.46) GRIK1CCR2KMT2AGAALMNA
SCHEMBL27614646 0.78 CA3 (0.42) KMT2ALMNANPC1RAB9ASMN1; SMN2
SCHEMBL1337289 0.76 IDO1 (0.41) GRIK1CCR2KMT2AGAALMNA
SCHEMBL28664691 0.76 CXCR2 (0.39) GRIK1CCR2KMT2AGAANPC1
Hydrochloric Acid SCHEMBL3641623 0.74 IDO1 (0.40) GRIK1CCR2KMT2AGAALMNA
SCHEMBL28172323 0.73 TP53 (0.48) KMT2AGAALMNANPC1HPGD
SCHEMBL12883495 0.71 CCR2 (0.42) GRIK1CCR2KMT2AGAALMNA
SCHEMBL12368470 0.71 NR4A2 (0.40) GRIK1CCR2KMT2AGAALMNA
SCHEMBL12895731 0.71 ALDH1A1 (0.40) GRIK1CCR2KMT2AGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2470526-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2012-07-04 EP disclosed
WO-2011025927-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2011-03-03 WO disclosed