SCHEMBL8214915

SCHEMBL8214915

N#Cc1ccc(NC(=O)NCS(=O)(=O)O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SAE1 Q9UBE0 1/20 0.58
UBA2 Q9UBT2 1/20 0.58
CA12 O43570 2/20 0.57
CA1 P00915 2/20 0.57
CA2 P00918 2/20 0.57
CA9 Q16790 2/20 0.57
MAPT P10636 3/20 0.55
LMNA P02545 2/20 0.55
TSHR P16473 1/20 0.55
HTT P42858 1/20 0.55
NLRP3 Q96P20 1/20 0.55
NAMPT P43490 7/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
KDM4E B2RXH2 1/20 0.54
POLB P06746 1/20 0.54
PKM P14618 1/20 0.54
MAPK1 P28482 1/20 0.54
RAB9A P51151 1/20 0.54
IL18 Q14116 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11050029 0.81 CNR1 (0.63) SAE1UBA2CA12CA1CA2
SCHEMBL11054945 0.79 MAPT (0.81) SAE1UBA2CA12CA1CA2
SCHEMBL23328727 0.79 RAB9A (0.60) CA12CA1CA2CA9MAPT
SCHEMBL25840768 0.79 NPC1 (0.60) CA12CA1CA2CA9NAMPT
SCHEMBL23329075 0.79 SAE1 (0.50) SAE1UBA2CA12CA1CA2
SCHEMBL11052863 0.79 SAE1 (0.63) SAE1UBA2CA12CA1CA2
SCHEMBL23328367 0.78 ACP1 (0.59) CA12CA1CA2CA9LMNA
SCHEMBL23329073 0.77 CA2 (0.53) CA12CA1CA2CA9MAPT
SCHEMBL8576539 0.76 CNR1 (0.66) SAE1UBA2CA12CA1CA2
SCHEMBL18054897 0.76 CNR1 (0.62) SAE1UBA2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6015792-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 2000-01-18 US disclosed
US-6008250-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 1999-12-28 US disclosed
US-5866608-A AROMATIC COMPOUNDS BIORESEARCH, INC. (US) 1999-02-02 US disclosed
US-5703053-A TASTELESS INGESTIBLE COMPOUNDS WHICH REDUCE OR ELIMINATE UNDESIRABLE TASTES IN EATABLES BIORESEARCH, INC. (US) 1997-12-30 US disclosed
US-5700792-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 1997-12-23 US disclosed
US-5665755-A NAPHTHO(1,2-D)IMIDAZOLE-5-SULFONATES (TASTANDS) USED TO REDUCE BITTER OR METALLIC TASTES; FOODS, DRUGS, ARTIFICIAL SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH INC. (US) 1997-09-09 US disclosed
US-5654311-A TASTANDS OF PYRIMIDINE DERIVATIVES, E.G. OROTIC ACID, TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH INC. (US) 1997-08-05 US disclosed
US-5650403-A PURINE-BASED COMPOUNDS (TASTANDS, E.G. IOSINE, GUANOSINE AND XANTHINE-5'-PHOSPHATE) USED TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; ARTIFICIAL SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-07-22 US disclosed
US-5646122-A COMPOUNDS (TASTANDS, E.G. A DIPEPTIDE CONTAINING TAURINE AND/OR ALANINE) USED TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; ARTIFICIAL SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-07-08 US disclosed
US-5643941-A PYRAN, THIOPYRAN AND CYCLOHEXANE DERIVATIVES (E.G. GLYCOSIDES AND INOSITOL, QUERCITOL) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS, DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-07-01 US disclosed
US-5631038-A COMPOUNDS (TASTANDS) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE ARE ADDED TO FOODS CONTAINING SODIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
EP-0661932-A4 SPECIFIC EATABLE TASTE MODIFIERS. BIORESEARCH INC (US) 1996-06-05 EP disclosed
EP-0661932-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1995-07-12 EP disclosed
EP-0417256-B1 NOVEL N-(SULFOMETHYL)-N'-ARYLUREAS NUTRASWEET CO (US) 1994-04-06 EP disclosed
US-5266717-A Suppressors of sweet and/or bitter tastes, adjuvants for foods or drugs NUTRASWEET PROPERTY HOLDINGS, INC. 1993-11-30 US disclosed
WO-1993010677-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1993-06-10 WO disclosed
EP-0417256-A4 NOVEL N-(SULFOMETHYL)-N'-ARYLUREAS 1991-09-25 EP disclosed
EP-0417256-A1 NOVEL N-(SULFOMETHYL)-N'-ARYLUREAS. NUTRASWEET CO (US) 1991-03-20 EP disclosed
US-4994490-A To inhibit or lessen sweet or bitter tastes in foods, beverage or drugs THE NUTRASWEET COMPANY (US) 1991-02-19 US disclosed
WO-1990011695-A1 NOVEL N-(SULFOMETHYL)-N'-ARYLUREAS THE NUTRASWEET COMPANY (US) 1990-10-18 WO disclosed