SCHEMBL8216183

SCHEMBL8216183

COCc1cccc(-c2cccc(COC)c2COC)c1COC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.42
KCNN4 O15554 1/20 0.34
HTT P42858 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALOX12 P18054 1/20 0.33
RAB9A P51151 1/20 0.33
IDO1 P14902 3/20 0.32
PRKCE Q02156 2/20 0.32
MYLK Q15746 2/20 0.32
MEN1 O00255 2/20 0.32
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 2/20 0.32
PRKCG P05129 1/20 0.32
MAPT P10636 1/20 0.32
PRKCA P17252 1/20 0.32
APEX1 P27695 1/20 0.32
RECQL P46063 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4962884 0.88 PDK2 (0.39) PDK2HTTNPSR1KDM4ENPC1
SCHEMBL49965 0.86 CD274 (0.46) PDK2KMT2APDCD1CD274
SCHEMBL1835122 0.78 PRKCE (0.42) PDK2HTTNPSR1KDM4ENPC1
SCHEMBL14954170 0.78 ALDH1A1 (0.42) PDK2HTTNPSR1KDM4ENPC1
SCHEMBL734879 0.78 KCNN4 (0.46) PDK2KCNN4HTTNPSR1KDM4E
SCHEMBL16245089 0.77 CD274 (0.44) PDK2KCNN4PDCD1CD274
SCHEMBL3931388 0.77 KDM4E (0.37) PDK2KDM4EIDO1CD274
Fluoride SCHEMBL1335703 0.77 PDK2 (0.33) PDK2HTTNPSR1KDM4ENPC1
SCHEMBL914993 0.76 PDK2 (0.38) PDK2HTTNPSR1KDM4ENPC1
SCHEMBL1666891 0.76 PDK2 (0.32) PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080587-A RATIONALLY DESIGNED LIBRARIES OF STRUCTURALLY-DIVERSE LOW MOLECULAR WEIGHT COMPOUNDS ELI LILLY AND COMPANY (US) 2000-06-27 US disclosed
EP-0712493-A4 A METHOD FOR PREPARING AND SELECTING PHARMACEUTICALLY USEFUL NON-PEPTIDE COMPOUNDS FROM A STRUCTURALLY DIVERSE UNIVERSAL LIBRARY SPHINX PHARMA CORP (US) 1997-01-15 EP disclosed
EP-0712493-A1 A METHOD FOR PREPARING AND SELECTING PHARMACEUTICALLY USEFUL NON-PEPTIDE COMPOUNDS FROM A STRUCTURALLY DIVERSE UNIVERSAL LIBRARY SPHINX PHARMACEUTICALS CORPORATION (US) 1996-05-22 EP disclosed
WO-1995004277-A1 A METHOD FOR PREPARING AND SELECTING PHARMACEUTICALLY USEFUL NON-PEPTIDE COMPOUNDS FROM A STRUCTURALLY DIVERSE UNIVERSAL LIBRARY SPHINX PHARMACEUTICALS CORPORATION (US) 1995-02-09 WO disclosed