SCHEMBL8216362

SCHEMBL8216362

COc1cc(-n2ccc(C(F)(F)F)n2)ccc1Br

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.49
MAPT P10636 5/20 0.49
RAB9A P51151 4/20 0.49
NPSR1 Q6W5P4 3/20 0.49
KDM4E B2RXH2 1/20 0.49
PTGS2 P35354 5/20 0.40
CCR1 P32246 1/20 0.40
HTT P42858 1/20 0.40
PAX8 Q06710 1/20 0.40
PTGS1 P23219 3/20 0.38
PRMT6 Q96LA8 1/20 0.38
POLB P06746 2/20 0.38
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16911209 0.83 NPC1 (0.49) NPC1MAPTRAB9ANPSR1KDM4E
SCHEMBL8201676 0.82 MAPT (0.48) NPC1MAPTRAB9ANPSR1KDM4E
SCHEMBL15476076 0.79 SUV39H2 (0.40) NPC1MAPTRAB9ANPSR1POLB
SCHEMBL24051557 0.78 NPC1 (0.44) NPC1MAPTRAB9ANPSR1KDM4E
SCHEMBL31110406 0.78 NPC1 (0.44) NPC1MAPTRAB9ANPSR1KDM4E
SCHEMBL12988881 0.77 PTGS2 (0.52) NPC1MAPTRAB9ANPSR1KDM4E
SCHEMBL15876687 0.77 ABCB11 (0.38) NPC1MAPTRAB9ANPSR1KDM4E
SCHEMBL3216783 0.77 NPC1 (0.44) NPC1MAPTRAB9ANPSR1KDM4E
SCHEMBL27588789 0.77 NOTUM (0.51) NPC1MAPTRAB9ANPSR1KDM4E
SCHEMBL15876568 0.76 ELOVL1 (0.43) NPC1MAPTRAB9ANPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed