SCHEMBL8218486

SCHEMBL8218486

O=C1Cc2ccc(-c3cccs3)cc2C1=O

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A11 P48066 1/20 0.52
BCHE P06276 1/20 0.44
CES1 P23141 1/20 0.44
KCNH2 Q12809 1/20 0.44
PGR P06401 2/20 0.42
ADORA1 P30542 1/20 0.41
SRD5A1 P18405 1/20 0.41
ERN1 O75460 1/20 0.41
PDK2 Q15119 1/20 0.40
PRMT6 Q96LA8 1/20 0.38
LTA4H P09960 1/20 0.38
HDAC3 O15379 3/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC2 Q92769 3/20 0.37
PRKDC P78527 2/20 0.37
ALOX5 P09917 1/20 0.36
CHEK1 O14757 1/20 0.36
CHEK2 O96017 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31358816 0.78 ADORA1 (0.55) SLC6A11KCNH2PGRADORA1SRD5A1
SCHEMBL2238249 0.78 ADORA1 (0.55) SLC6A11KCNH2PGRADORA1SRD5A1
SCHEMBL4243227 0.77 SLC6A11 (0.48) SLC6A11KCNH2PGRADORA1SRD5A1
SCHEMBL30512416 0.76 SLC6A11 (0.61) SLC6A11KCNH2PGRERN1PDK2
SCHEMBL21580251 0.76 SLC6A11 (0.61) SLC6A11KCNH2PGRERN1PDK2
SCHEMBL14322894 0.76 PDK2 (0.52) SLC6A11KCNH2ADORA1ERN1PDK2
SCHEMBL15571040 0.74 CLK4 (0.60) SLC6A11KCNH2PGRERN1PDK2
SCHEMBL27554974 0.73 SLC6A11 (0.58) SLC6A11KCNH2PGRADORA1ERN1
SCHEMBL3460160 0.73 HSD17B1 (0.53) SLC6A11KCNH2PGRADORA1SRD5A1
SCHEMBL8214476 0.73 PTPRC (0.54) BCHECES1KCNH2ERN1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127189-A CONTACTING WITH A 1,2-INDANEDIONE DERIVATIVE, MEASURING ABSORBANCE OR FLUORESCENCE OF PRODUCT FORMED, AND COMPARING TO STANDARDS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2000-10-03 US claimed
WO-1998020344-A1 COMPOSITIONS AND METHODS FOR DETECTION OF AN AMINE COMPOUND THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-05-14 WO claimed
US-6127189-A CONTACTING WITH A 1,2-INDANEDIONE DERIVATIVE, MEASURING ABSORBANCE OR FLUORESCENCE OF PRODUCT FORMED, AND COMPARING TO STANDARDS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2000-10-03 US disclosed
WO-1998020344-A1 COMPOSITIONS AND METHODS FOR DETECTION OF AN AMINE COMPOUND THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-05-14 WO disclosed