SCHEMBL8220809

SCHEMBL8220809

COc1cn[nH]c(=O)c1-c1cccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
HPGD P15428 3/20 0.50
KDM4E B2RXH2 2/20 0.50
MAPT P10636 3/20 0.48
MEN1 O00255 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD17B10 Q99714 3/20 0.47
PARP1 P09874 1/20 0.47
PRKCI P41743 1/20 0.47
PDE4B Q07343 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PDGFRB P09619 1/20 0.46
STK10 O94804 1/20 0.43
SLK Q9H2G2 1/20 0.43
MAPK1 P28482 1/20 0.43
TYMP P19971 1/20 0.43
GAA P10253 1/20 0.42
ALOX15 P16050 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8219871 0.81 ALDH1A1 (0.54) ALDH1A1KDM4EHSD17B10PARP1PRKCI
SCHEMBL34473210 0.80 KMT2A (0.46) ALDH1A1HPGDKDM4EMAPTMEN1
SCHEMBL8212270 0.79 ALDH1A1 (0.49) ALDH1A1HPGDKDM4EMAPTMEN1
SCHEMBL7796061 0.73 MAPT (0.63) ALDH1A1HPGDKDM4EMAPTMEN1
SCHEMBL20406100 0.71 ALDH1A1 (0.47) ALDH1A1HPGDKDM4EMAPTMEN1
SCHEMBL24861080 0.71 ALDH1A1 (0.59) ALDH1A1HPGDKDM4ESMN1; SMN2HSD17B10
SCHEMBL13323912 0.71 MAPT (0.44) ALDH1A1KDM4EMAPTMEN1RAB9A
SCHEMBL8220603 0.71 ALDH1A1 (0.53) ALDH1A1KDM4EHSD17B10PARP1PRKCI
SCHEMBL12880138 0.71 MAPT (0.75) ALDH1A1HPGDKDM4EMAPTMEN1
SCHEMBL29512056 0.71 MAPT (0.75) ALDH1A1HPGDKDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008019303-A2 PYRIDAZINONYL MACROCYCLIC HEPATITIS C SERINE PROTEASE INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed