SCHEMBL8219871

SCHEMBL8219871

O=c1[nH]ncc(-c2cccc3ccccc23)c1-c1cccc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
PARP1 P09874 1/20 0.54
PRKCI P41743 1/20 0.54
PDE4B Q07343 1/20 0.54
HSD17B10 Q99714 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
TYMP P19971 1/20 0.48
KDM4E B2RXH2 1/20 0.41
ALPL P05186 1/20 0.41
GAA P10253 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
NOS1 P29475 1/20 0.40
TRPM2 O94759 1/20 0.39
DHFR P00374 1/20 0.39
PDE10A Q9Y233 1/20 0.39
MAPK1 P28482 1/20 0.39
PTPN1 P18031 1/20 0.38
KCNQ3 O43525 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8220603 0.83 ALDH1A1 (0.53) ALDH1A1PARP1PRKCIPDE4BHSD17B10
SCHEMBL8220809 0.81 ALDH1A1 (0.50) ALDH1A1PARP1PRKCIPDE4BHSD17B10
SCHEMBL8212270 0.79 ALDH1A1 (0.49) ALDH1A1PARP1PRKCIPDE4BHSD17B10
SCHEMBL8220691 0.79 ALDH1A1 (0.49) ALDH1A1PARP1PRKCIPDE4BHSD17B10
SCHEMBL8219861 0.79 ALDH1A1 (0.49) ALDH1A1PARP1PRKCIPDE4BHSD17B10
SCHEMBL8220600 0.76 ALDH1A1 (0.45) ALDH1A1PARP1PRKCIPDE4BHSD17B10
SCHEMBL21514162 0.73 METAP2 (0.66) ALDH1A1PARP1PRKCIPDE4BHSD17B10
SCHEMBL24087861 0.72 CYP1A2 (0.57) ALDH1A1PARP1PRKCIPDE4BHSD17B10
Phthalazinone SCHEMBL51553 0.71 PARP1 (1.00) ALDH1A1PARP1PRKCIPDE4BHSD17B10
SCHEMBL577268 0.71 KDM4E (0.49) ALDH1A1PARP1PRKCIPDE4BHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008019303-A2 PYRIDAZINONYL MACROCYCLIC HEPATITIS C SERINE PROTEASE INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed