SCHEMBL8220976

SCHEMBL8220976

O=C(c1ccc2oc(NCc3cccc(Cl)c3)nc2c1)N(Cc1cccnc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
THRB P10828 4/20 0.52
PDK1 Q15118 5/20 0.49
GAA P10253 2/20 0.47
TSHR P16473 1/20 0.47
HDAC6 Q9UBN7 3/20 0.46
HDAC1 Q13547 1/20 0.46
TP53 P04637 2/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8219821 0.86 THRB (0.60) THRBHDAC6HDAC1TP53
SCHEMBL8226183 0.85 THRB (0.66) THRBPDK1HDAC6HDAC1NPC1
SCHEMBL8225281 0.85 THRB (0.56) THRBPDK1HDAC6HDAC1NPC1
SCHEMBL8229490 0.84 THRB (0.55) THRBPDK1HDAC6HDAC1NPC1
SCHEMBL8228581 0.83 THRB (0.59) THRBHDAC6HDAC1NPC1MAPT
SCHEMBL8229448 0.83 THRB (0.59) THRBPDK1HDAC6HDAC1NPC1
SCHEMBL8231039 0.80 THRB (0.56) THRBGAATSHRKMT2A
SCHEMBL5364592 0.80 THRB (0.57) THRBGAAHDAC6HDAC1MEN1
SCHEMBL8228557 0.77 THRB (0.58) THRBHDAC6HDAC1
SCHEMBL8219815 0.77 THRB (0.61) THRBHDAC6HDAC1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007140982-A1 SUBSTITUTED BENZOXAZOLES BAYER HEALTHCARE AG (DE) 2007-12-13 WO disclosed