SCHEMBL8222575

SCHEMBL8222575

Nc1ccccc1C1(O)CCNCC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.57
DRD2 P14416 2/20 0.43
OPRM1 P35372 4/20 0.40
HTR2A P28223 3/20 0.37
SLC6A2 P23975 1/20 0.37
HTR2C P28335 1/20 0.37
SLC6A4 P31645 1/20 0.37
DPP9 Q86TI2 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
TSHR P16473 2/20 0.34
OPRL1 P41146 3/20 0.34
OPRD1 P41143 2/20 0.34
OPRK1 P41145 2/20 0.34
PDK2 Q15119 1/20 0.34
BACE1 P56817 1/20 0.34
CYP3A4 P08684 2/20 0.33
USP2 O75604 2/20 0.33
CYP2D6 P10635 2/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2079404 0.86 ALOX15 (0.41) SIGMAR1OPRM1TSHROPRL1OPRD1
SCHEMBL29710660 0.82 ALOX15 (0.38) SIGMAR1OPRM1TSHROPRL1OPRD1
SCHEMBL1703171 0.82 ALOX15 (0.38) SIGMAR1OPRM1TSHROPRL1OPRD1
SCHEMBL7102084 0.82 ALOX15 (0.38) SIGMAR1OPRM1TSHROPRL1OPRD1
SCHEMBL1660350 0.82 SIGMAR1 (0.62) SIGMAR1DRD2OPRM1HTR2ASLC6A2
SCHEMBL2270935 0.81 SIGMAR1 (0.62) SIGMAR1DRD2OPRM1HTR2COPRL1
Hydrochloric Acid SCHEMBL10007651 0.80 SIGMAR1 (0.61) SIGMAR1DRD2OPRM1HTR2ASLC6A2
SCHEMBL632646 0.80 OPRM1 (0.37) SIGMAR1OPRM1SLC6A2SLC6A4OPRL1
SCHEMBL7101793 0.80 OPRM1 (0.37) SIGMAR1OPRM1SLC6A2SLC6A4OPRL1
Hydrochloric Acid SCHEMBL8175707 0.79 SIGMAR1 (0.60) SIGMAR1DRD2OPRM1HTR2COPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021375-A2 MODULATORS OF MUSCARINIC RECEPTORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-02-21 WO disclosed