SCHEMBL8223286

SCHEMBL8223286

CC1=C(C(=O)O)C(c2c(C)cccc2I)C(C2OC(C)O2)=C(C)N1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 5/20 0.33
ALDH1A1 P00352 2/20 0.31
MAPT P10636 2/20 0.31
KDM4E B2RXH2 3/20 0.30
NPSR1 Q6W5P4 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8224837 0.81 CACNA1B (0.32) CACNA1BALDH1A1MAPTKDM4ENPSR1
SCHEMBL8224820 0.76 CACNA1B (0.35) CACNA1BALDH1A1MAPTKDM4ECYP1A2
SCHEMBL8224367 0.75 CACNA1B (0.35) CACNA1BALDH1A1MAPTKDM4ENPSR1
SCHEMBL8218968 0.75 CACNA1B (0.35) CACNA1BALDH1A1MAPTKDM4ENPSR1
SCHEMBL8222248 0.74 GAA (0.43) CACNA1BALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL8222271 0.70 KDM4E (0.48) ALDH1A1MAPTKDM4ENPSR1CYP1A2
SCHEMBL8225580 0.68 KDM4E (0.54) ALDH1A1MAPTKDM4ENPSR1CYP1A2
SCHEMBL8298006 0.64 CACNA1B (0.40) CACNA1BALDH1A1MAPTKDM4ECYP1A2
SCHEMBL27544295 0.63 TSHR (0.46) CACNA1BALDH1A1MAPTKDM4ENPSR1
SCHEMBL8222581 0.63 KDM4E (0.48) CACNA1BALDH1A1MAPTKDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008006070-A2 COMPOUNDS AND COMBINATIONS THEREOF FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF USE THEREOF ROSKAMP RESEARCH LLC (US) 2008-01-10 WO disclosed