SCHEMBL8224837

SCHEMBL8224837

CC1=C(C(=O)O)C(c2cccc(C)c2C)C(C2OC(C)O2)=C(C)N1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 8/20 0.32
CCR2 P41597 1/20 0.32
HTR2C P28335 3/20 0.32
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2B P41595 1/20 0.32
GAA P10253 2/20 0.32
MGAM O43451 1/20 0.32
AMY1A P0DUB6 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
KDM4E B2RXH2 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
MGLL Q99685 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8218968 0.84 CACNA1B (0.35) CACNA1BCCR2HTR2CMAPTALDH1A1
SCHEMBL8224367 0.84 CACNA1B (0.35) CACNA1BCCR2HTR2CMAPTALDH1A1
SCHEMBL8222248 0.83 GAA (0.43) CACNA1BALDH1A1GAAKDM4ECYP1A2
SCHEMBL8224820 0.83 CACNA1B (0.35) CACNA1BMAPTALDH1A1GAAKDM4E
SCHEMBL8223286 0.81 CACNA1B (0.33) CACNA1BMAPTALDH1A1GAAKDM4E
SCHEMBL8222581 0.71 KDM4E (0.48) CACNA1BCCR2HTR2CMAPTALDH1A1
SCHEMBL27544295 0.71 TSHR (0.46) CACNA1BCCR2HTR2CMAPTALDH1A1
SCHEMBL8222583 0.71 KDM4E (0.52) CACNA1BCCR2HTR2CMAPTALDH1A1
SCHEMBL8222269 0.70 GAA (0.47) MAPTALDH1A1GAAMGAMAMY1A
SCHEMBL8222265 0.70 KDM4E (0.68) HTR2CMAPTALDH1A1HTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008006070-A2 COMPOUNDS AND COMBINATIONS THEREOF FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF USE THEREOF ROSKAMP RESEARCH LLC (US) 2008-01-10 WO disclosed