SCHEMBL8224367

SCHEMBL8224367

CC1=C(C(=O)O)C(c2ccccc2N)C(C2OC(C)O2)=C(C)N1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 13/20 0.35
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
ADORA3 P0DMS8 2/20 0.33
ABCC4 O15439 1/20 0.33
PLIN1 O60240 1/20 0.33
CACNA1F O60840 1/20 0.33
GMNN O75496 1/20 0.33
KCNK2 O95069 1/20 0.33
ABCB11 O95342 1/20 0.33
GSR P00390 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8218968 0.88 CACNA1B (0.35) CACNA1BKDM4EALDH1A1MAPTADORA3
SCHEMBL8222248 0.86 GAA (0.43) CACNA1BKDM4EALDH1A1TP53CYP1A2
SCHEMBL8224837 0.84 CACNA1B (0.32) CACNA1BKDM4EALDH1A1MAPTCYP1A2
SCHEMBL8224820 0.79 CACNA1B (0.35) CACNA1BKDM4EALDH1A1MAPTLMNA
SCHEMBL8223286 0.75 CACNA1B (0.33) CACNA1BKDM4EALDH1A1MAPTCYP1A2
SCHEMBL8222581 0.75 KDM4E (0.48) CACNA1BKDM4EALDH1A1MAPTADORA3
SCHEMBL8222583 0.74 KDM4E (0.52) CACNA1BKDM4EALDH1A1MAPTADORA3
SCHEMBL8225874 0.73 CACNA1F (0.51) KDM4EALDH1A1MAPTADORA3CACNA1F
SCHEMBL8222271 0.72 KDM4E (0.48) KDM4EALDH1A1MAPTADORA3CACNA1F
SCHEMBL8214725 0.72 KDM4E (0.55) KDM4EALDH1A1MAPTADORA3CACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008006070-A2 COMPOUNDS AND COMBINATIONS THEREOF FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF USE THEREOF ROSKAMP RESEARCH LLC (US) 2008-01-10 WO disclosed