SCHEMBL8226019

SCHEMBL8226019

NC(=O)c1n[nH]cc1NC(=O)NCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CFD P00746 1/20 0.51
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.50
IKBKB O14920 1/20 0.50
GSK3B P49841 1/20 0.50
GAA P10253 1/20 0.50
POLB P06746 2/20 0.49
ROCK2 O75116 2/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
MMP3 P08254 1/20 0.47
CA2 P00918 4/20 0.46
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA9 Q16790 3/20 0.46
HTT P42858 1/20 0.45
LMNA P02545 1/20 0.44
ROCK1 Q13464 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8220657 0.77 EPHX1 (0.46) CFDKDM4EALDH1A1GSK3BGAA
SCHEMBL12000436 0.77 EPHX1 (0.46) CFDKDM4EALDH1A1GSK3BGAA
SCHEMBL6470700 0.76 IKBKB (0.36) KDM4EALDH1A1IKBKBGAA
SCHEMBL5274230 0.76 HPGD (0.49) ALDH1A1GSK3BGAAROCK2HDAC1
SCHEMBL5274499 0.75 KMT2A (0.46) KDM4EALDH1A1GAAPOLBHTT
SCHEMBL5267185 0.73 POLB (0.48) KDM4EALDH1A1GAAPOLBROCK2
SCHEMBL13816854 0.73 ALDH1A1 (0.50) KDM4EALDH1A1GAAPOLB
SCHEMBL1709275 0.73 CFD (0.57) CFDKDM4EALDH1A1GSK3BGAA
SCHEMBL5269714 0.73 ROCK2 (0.54) GSK3BROCK2HDAC1HDAC6ROCK1
SCHEMBL5270571 0.73 KMT2A (0.59) ALDH1A1GAAPOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008007113-A2 PHARMACEUTICAL COMBINATIONS ASTEX THERAPEUTICS LIMITED (GB) 2008-01-17 WO disclosed