SCHEMBL8226157

SCHEMBL8226157

O=C(NC1CCCCC1)c1ccc(Cn2ccnc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.57
RAB9A P51151 3/20 0.57
KMT2A Q03164 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
KDM4E B2RXH2 1/20 0.55
CYP19A1 P11511 4/20 0.54
NAMPT P43490 2/20 0.53
TBXAS1 P24557 2/20 0.51
POLB P06746 1/20 0.51
CYP1A2 P05177 1/20 0.50
HPGD P15428 1/20 0.50
CYP2C19 P33261 1/20 0.50
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8738903 0.81 EZH2 (0.53) NPC1KMT2ACYP19A1TBXAS1POLB
SCHEMBL26401026 0.79 KMT2A (0.71) NPC1RAB9AKMT2ASMN1; SMN2NAMPT
SCHEMBL8810497 0.78 HRH3 (0.54) KDM4ECYP19A1TBXAS1POLBCYP1A2
SCHEMBL7879609 0.77 GAA (0.53) NPC1KMT2ASMN1; SMN2KDM4ECYP19A1
SCHEMBL7875125 0.76 KMT2A (0.43) NPC1RAB9AKMT2ASMN1; SMN2NAMPT
SCHEMBL506708 0.76 NPC1 (0.64) NPC1RAB9AKMT2ASMN1; SMN2KDM4E
SCHEMBL126657 0.75 NPC1 (0.82) NPC1RAB9AKMT2ASMN1; SMN2CYP1A2
SCHEMBL520877 0.75 NPC1 (0.82) NPC1RAB9AKMT2ASMN1; SMN2CYP1A2
SCHEMBL28928584 0.75 NPC1 (0.82) NPC1RAB9AKMT2ASMN1; SMN2CYP1A2
SCHEMBL4492287 0.74 CYP19A1 (0.75) KMT2ACYP19A1TBXAS1POLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028942-A2 DIPEPTIDE NITRILES Novartis AG (CH) 2000-08-23 EP disclosed
WO-1999024460-A2 DIPEPTIDE NITRILES NOVARTIS AG (CH) 1999-05-20 WO disclosed